SCHEMBL4078733

SCHEMBL4078733

CCCOC(=O)c1cc2c(o1)c(NC(=O)c1ccc(C#N)cc1)nn2C(=O)OCC

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
KDM4E B2RXH2 2/20 0.44
ELANE P08246 1/20 0.40
PKM P14618 2/20 0.39
P2RY14 Q15391 1/20 0.38
GPR35 Q9HC97 2/20 0.37
ITK Q08881 3/20 0.37
POLB P06746 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
BTK Q06187 1/20 0.36
MAPT P10636 3/20 0.35
LMNA P02545 2/20 0.35
TSHR P16473 1/20 0.35
BRAF P15056 1/20 0.35
MAPK14 Q16539 1/20 0.35
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4091779 0.88 LMNA (0.44) ALDH1A1SMN1; SMN2KDM4EELANEP2RY14
SCHEMBL4088637 0.88 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2KDM4EELANEGPR35
SCHEMBL4078418 0.88 HTT (0.43) ALDH1A1SMN1; SMN2KDM4EELANEMAPT
SCHEMBL4083509 0.88 GPR35 (0.49) ALDH1A1SMN1; SMN2KDM4EELANEGPR35
SCHEMBL4088619 0.85 GPR35 (0.42) ALDH1A1ELANEGPR35MAPTMAPK14
SCHEMBL4083134 0.85 GPR35 (0.42) ALDH1A1SMN1; SMN2KDM4EELANEGPR35
SCHEMBL4084033 0.84 ELANE (0.45) ALDH1A1ELANEGPR35LMNATSHR
SCHEMBL4083252 0.84 PTK2 (0.37) ALDH1A1SMN1; SMN2KDM4EELANEGPR35
SCHEMBL4086291 0.84 MAPK1 (0.44) SMN1; SMN2KDM4EPOLBMAPTLMNA
SCHEMBL4091205 0.84 LRRK2 (0.46) ALDH1A1SMN1; SMN2KDM4EPKMBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed