SCHEMBL4083134

SCHEMBL4083134

CCCOC(=O)c1cc2c(o1)c(NC(=O)c1ccc(OC(F)(F)F)cc1)nn2C(=O)OCC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 1/20 0.42
MAPT P10636 1/20 0.41
EPHX2 P34913 1/20 0.39
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
ALDH1A1 P00352 4/20 0.38
HPGD P15428 4/20 0.38
KDM4E B2RXH2 3/20 0.38
GAA P10253 1/20 0.38
ELANE P08246 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
CYP2C9 P11712 3/20 0.38
CYP2C19 P33261 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TRPV1 Q8NER1 2/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083509 0.90 GPR35 (0.49) GPR35MAPTALDH1A1HPGDKDM4E
SCHEMBL4091779 0.89 LMNA (0.44) GPR35MAPTALDH1A1HPGDKDM4E
SCHEMBL4088619 0.88 GPR35 (0.42) GPR35MAPTPPARGPPARAALDH1A1
SCHEMBL4088637 0.88 ALDH1A1 (0.43) GPR35MAPTALDH1A1HPGDKDM4E
SCHEMBL4078418 0.87 HTT (0.43) MAPTALDH1A1HPGDKDM4EGAA
SCHEMBL4078733 0.85 ALDH1A1 (0.44) GPR35MAPTALDH1A1KDM4EELANE
SCHEMBL4082122 0.84 MCHR1 (0.42) MAPTALDH1A1KDM4EHDAC1
SCHEMBL4078227 0.83 PAX8 (0.45) GPR35MAPTALDH1A1KDM4EGAA
SCHEMBL4084033 0.83 ELANE (0.45) GPR35ALDH1A1ELANENPC1
SCHEMBL4083252 0.83 PTK2 (0.37) GPR35MAPTALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP claimed
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed