SCHEMBL4083862

SCHEMBL4083862

CCCOC(=O)c1cc2c(o1)c(NC(=O)c1cc(C)c(C)o1)nn2C(=O)OCC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
RAB9A P51151 8/20 0.37
NPC1 O15118 7/20 0.37
SMN1; SMN2 Q16637 6/20 0.37
ALDH1A1 P00352 6/20 0.37
HPGD P15428 4/20 0.37
TP53 P04637 4/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
THRB P10828 2/20 0.34
MITF O75030 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
MAOB P27338 1/20 0.33
MAPK1 P28482 1/20 0.33
AKR1C3 P42330 1/20 0.33
HSP90AA1 P07900 2/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4084026 0.86 MAPT (0.42) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL4087183 0.85 RAB9A (0.45) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL4078418 0.85 HTT (0.43) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL4084062 0.84 ALDH1A1 (0.51) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL4084041 0.84 RAB9A (0.45) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL4088615 0.84 KMT2A (0.45) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL4093521 0.83 SMN1; SMN2 (0.43) TAS1R3TAS1R1RAB9ANPC1SMN1; SMN2
SCHEMBL4091779 0.83 LMNA (0.44) RAB9ASMN1; SMN2ALDH1A1HPGDKMT2A
SCHEMBL4081200 0.83 MAPT (0.45) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD
SCHEMBL4087974 0.83 TAS2R8 (0.35) RAB9ANPC1SMN1; SMN2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed