Phenazepam

Phenazepam

SCHEMBL416137

O=C1CN=C(c2ccccc2Cl)c2cc(Br)ccc2N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 6/20 1.00
GABRA5 P31644 6/20 1.00
GABRA3 P34903 6/20 1.00
GABRA2 P47869 6/20 1.00
GABRB2 P47870 5/20 1.00
GABRG2 P18507 4/20 0.77
GABRB3 P28472 4/20 0.77
GABRP O00591 3/20 0.77
GABRD O14764 3/20 0.77
GABRB1 P18505 3/20 0.77
GABRA4 P48169 3/20 0.77
GABRE P78334 3/20 0.77
GABRA6 Q16445 3/20 0.77
GABRG1 Q8N1C3 3/20 0.77
GABRG3 Q99928 3/20 0.77
GABRQ Q9UN88 3/20 0.77
ADRA1A P35348 2/20 0.67
KMT2A Q03164 2/20 0.65
LMNA P02545 1/20 0.59
CNR1 P21554 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenazepam SCHEMBL29368536 1.00 GABRA1 (1.00) GABRA1GABRA5GABRA3GABRA2GABRB2
Delorazepam SCHEMBL157332 0.87 GABRA1 (1.00) GABRA1GABRA5GABRA3GABRA2GABRB2
Delorazepam SCHEMBL32681132 0.87 GABRA1 (1.00) GABRA1GABRA5GABRA3GABRA2GABRB2
Delorazepam SCHEMBL29375434 0.87 GABRA1 (1.00) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL18166494 0.87 GABRA1 (0.77) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL7720989 0.85 GABRA1 (0.77) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL16144652 0.85 GABRA1 (0.77) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL9378946 0.85 GABRA1 (0.77) GABRA1GABRA5GABRA3GABRA2GABRB2
7-Aminoclonazepam SCHEMBL11453747 0.85 GABRA1 (0.77) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL11772087 0.85 GABRA1 (0.77) GABRA1GABRA5GABRA3GABRA2GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 743 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3507371-B1 COMPOSITIONS FOR TREATING DISEASES AND DISORDERS OF THE NERVOUS SYSTEM UNIV RUTGERS (US) 2026-01-28 EP claimed
US-20230174613-A1 METHODS AND COMPOSITIONS FOR TREATING DISEASES AND DISORDERS OF THE NERVOUS SYSTEM RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2023-06-08 US claimed
US-11542315-B2 Methods and compositions for treating diseases and disorders of the nervous system RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2023-01-03 US claimed
US-11510929-B2 Mitigation of epileptic seizures by combination therapy using benzodiazepines and neurosteroids THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-11-29 US claimed
US-20200316087-A1 NOVEL COMBINATION THERAPY FOR ANXIETY DISORDERS, EPILEPSY, AND PAIN THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK 2020-10-08 US claimed
US-20200215078-A1 MITIGATION OF EPILEPTIC SEIZURES BY COMBINATION THERAPY USING BENZODIAZEPINES AND NEUROSTEROIDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-07-09 US claimed
US-20200030304-A1 MITIGATION OF CNS DISORDERS BY COMBINATION THERAPY USING NEUROSTEROIDS, AND AMPA BLOCKERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-01-30 US claimed
US-10426786-B2 Mitigation of epileptic seizures by combination therapy using benzodiazepines and neurosteroids THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-10-01 US claimed
EP-3507371-A1 METHODS AND COMPOSITIONS FOR TREATING DISEASES AND DISORDERS OF THE NERVOUS SYSTEM Rutgers, The State University of New Jersey (US) 2019-07-10 EP claimed
US-20190194287-A1 METHODS AND COMPOSITIONS FOR TREATING DISEASES AND DISORDERS OF THE NERVOUS SYSTEM RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2019-06-27 US claimed
US-20130309306-A1 INTRAPULMONARY BENZODIAZEPINE FOR THE TREATMENT AND PREVENTION OF SEIZURES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-11-21 US claimed
EP-2649443-A2 METHODS AND KITS FOR DETECTION OF DRUGS Ramot at Tel-Aviv University Ltd (IL) 2013-10-16 EP claimed
CN-103354902-A Drug detection method and kit UNIV RAMOT 2013-10-16 CN claimed
WO-2013096560-A1 EXCIPIENT-FREE AEROSOL FORMULATION MAP PHARMACEUTICALS, INC. (US) 2013-06-27 WO claimed
US-20130156823-A1 Excipient-free Aerosol Formulation MAP Pharmacauticals, Inc. (US) 2013-06-20 US claimed
WO-2012077110-A2 METHODS AND KITS FOR DETECTION OF DRUGS RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2012-06-14 WO claimed
WO-2012075286-A2 INTRAPULMONARY BENZODIAZEPINE FOR THE TREATMENT AND PREVENTION OF SEIZURES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-06-07 WO claimed
WO-2012071220-A1 COMPOSITIONS AND METHODS FOR ONCE-DAILY ADMINISTRATION OF A TRILAYER OSMOTIC TABLET TRANSCEPT PHARMACEUTICALS, INC. (US) 2012-05-31 WO claimed
US-20120128778-A1 COMPOSITIONS AND METHODS FOR ONCE-DAILY ADMINISTRATION OF A TRILAYER OSMOTIC TABLET TRANSCEPT PHARMACEUTICALS, INC. 2012-05-24 US claimed
WO-2008033351-A2 MULTIMODAL ABUSE RESISTANT AND EXTENDED RELEASE FORMULATIONS THERAQUEST BIOSCIENCES, INC. (US) 2008-03-20 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11510929-B2 Mitigation of epileptic seizures by combination therapy using benzodiazepines and neurosteroids GABRB2, GABRA4, GABRB1 GABRA1 7/4885GABRA5 8/4885GABRA3 9/4885
US-20200030304-A1 MITIGATION OF CNS DISORDERS BY COMBINATION THERAPY USING NEUROSTEROIDS, AND AMPA BLOCKERS GABRA4, GABRG1, GABRB2 GABRA1 9/4885GABRA5 16/4885GABRA3 10/4885
US-10426786-B2 Mitigation of epileptic seizures by combination therapy using benzodiazepines and neurosteroids GABRB2, GABRA4, GABRB1 GABRA1 7/4885GABRA5 8/4885GABRA3 9/4885
US-20200316087-A1 NOVEL COMBINATION THERAPY FOR ANXIETY DISORDERS, EPILEPSY, AND PAIN GABRB2, GABRB1, GABRB3 GABRA1 5/4885GABRA5 15/4885GABRA3 7/4885
US-20200215078-A1 MITIGATION OF EPILEPTIC SEIZURES BY COMBINATION THERAPY USING BENZODIAZEPINES AND NEUROSTEROIDS GABRB2, GABRA4, GABRB1 GABRA1 7/4885GABRA5 8/4885GABRA3 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.