SCHEMBL4240804

SCHEMBL4240804

O=C1CC(c2ccccc2)NC(c2ccccc2)C1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.55
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
LMNA P02545 1/20 0.50
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
ALDH1A1 P00352 1/20 0.47
PRCP P42785 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13911781 1.00 SMN1; SMN2 (0.55) SMN1; SMN2MEN1KMT2ALMNAGAA
Hydrochloric Acid SCHEMBL28391104 0.98 SMN1; SMN2 (0.53) SMN1; SMN2MEN1KMT2ALMNAGAA
Ethylene SCHEMBL8557034 0.96 SMN1; SMN2 (0.51) SMN1; SMN2MEN1KMT2ALMNAGAA
SCHEMBL6984427 0.86 SMN1; SMN2 (0.56) SMN1; SMN2MEN1KMT2ALMNAGAA
SCHEMBL5738919 0.78 PRCP (0.60) SMN1; SMN2MEN1KMT2ALMNAGAA
SCHEMBL13911779 0.78 DDB1 (0.41) SMN1; SMN2MEN1KMT2ALMNAGAA
SCHEMBL6140740 0.78 PRCP (0.60) SMN1; SMN2MEN1KMT2ALMNAGAA
Ethylene SCHEMBL8554182 0.78 LMNA (0.45) SMN1; SMN2MEN1KMT2ALMNAGAA
SCHEMBL19283462 0.78 MEN1 (0.64) SMN1; SMN2MEN1KMT2ALMNAPRCP
SCHEMBL29413705 0.77 SMN1; SMN2 (0.40) SMN1; SMN2MEN1KMT2ALMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110963960-B Compound for promoting watermelon expansion and watermelon expansion liquid fertilizer 南京汉尔斯生物科技有限公司 2021-05-28 CN claimed
CN-110963960-A Compound for promoting watermelon expansion and watermelon expansion liquid fertilizer 南京汉尔斯生物科技有限公司 2020-04-07 CN claimed
CN-110963960-B Compound for promoting watermelon expansion and watermelon expansion liquid fertilizer 南京汉尔斯生物科技有限公司 2021-05-28 CN disclosed
CN-110963960-A Compound for promoting watermelon expansion and watermelon expansion liquid fertilizer 南京汉尔斯生物科技有限公司 2020-04-07 CN disclosed
US-9174960-B2 Compounds useful against kinetoplastideae parasites CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2015-11-03 US disclosed
US-9174960-B2 Compounds useful against kinetoplastideae parasites CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2015-11-03 US disclosed
EP-2664617-A1 Method of making a 2,6-diaryl piperidine derivative Genzyme Corporation (US) 2013-11-20 EP disclosed
US-20120214996-A1 COMPOUNDS USEFUL AGAINST KINETOPLASTIDEAE PARASITES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-08-23 US disclosed
US-20120214996-A1 COMPOUNDS USEFUL AGAINST KINETOPLASTIDEAE PARASITES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-08-23 US disclosed
WO-2011033115-A2 COMPOUNDS USEFUL AGAINST KINETOPLASTIDEAE PARASITES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2011-03-24 WO disclosed
US-7501518-B2 Methods of making 2,6-diaryl piperidine derivatives GENZYME CORPORATION (US) 2009-03-10 US disclosed
US-6420364-B1 TREATING AUTOIMMUNE DISEASES,ALZHEIMER'S DISEASE, ATHEROSCLEROSIS, OSTEOPOROSIS, BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-07-16 US disclosed
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
US-20020058809-A1 Compounds useful as reversible inhibitors of cysteine proteases EMMANUEL MICHEL JOSE (US) 2002-05-16 US disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed
EP-0567430-B1 Substituted 1-Hydroxy-2,6-Diaryl-4-Piperidone Ketal Stabilizers CIBA GEIGY AG (CH) 1998-02-18 EP disclosed
EP-0567430-A1 Substituted 1-Hydroxy-2,6-Diaryl-4-Piperidone Ketal Stabilizers CIBA-GEIGY AG (CH) 1993-10-27 EP disclosed
US-5235056-A Discoloration inhibitors CIBA-GEIGY CORPORATION (US) 1993-08-10 US disclosed
EP-0056699-B1 ORGANIC PEROXIDES AND USE OF SAME AUSIMONT S.p.A. (IT) 1986-04-09 EP disclosed
EP-0056699-A1 Organic peroxides and use of same AUSIMONT S.p.A. (IT) 1982-07-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020058809-A1 Compounds useful as reversible inhibitors of cysteine proteases CTSS, CTSK, CTSB SMN1; SMN2 4666/4885MEN1 3318/4885KMT2A 4513/4885
US-20120214996-A1 COMPOUNDS USEFUL AGAINST KINETOPLASTIDEAE PARASITES TST, PDXK, TBCB SMN1; SMN2 3140/4885MEN1 4710/4885KMT2A 962/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.