SCHEMBL4244760

SCHEMBL4244760

O=C(c1ccsc1)N(c1cccnc1)C1CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.47
OPRD1 P41143 2/20 0.47
OPRK1 P41145 2/20 0.47
CHRM3 P20309 1/20 0.45
SLC6A2 P23975 5/20 0.40
SLC6A4 P31645 5/20 0.40
SLC6A3 Q01959 5/20 0.40
CACNA2D1 P54289 2/20 0.36
TBXAS1 P24557 2/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
GPBAR1 Q8TDU6 1/20 0.36
KCNH2 Q12809 2/20 0.35
CYP2D6 P10635 1/20 0.34
CYP3A4 P08684 2/20 0.34
LCK P06239 1/20 0.34
FYN P06241 1/20 0.34
DAO P14920 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14349560 0.81 CHRM3 (0.51) CHRM3SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL14349504 0.79 TRPM8 (0.50) OPRM1OPRD1CHRM3SLC6A2SLC6A4
SCHEMBL10462601 0.78 OPRM1 (0.82) OPRM1OPRD1OPRK1CHRM3
SCHEMBL30502020 0.72 GPR119 (0.40) CHRM3SLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL3662258 0.71 SLC6A2 (0.44) CHRM3SLC6A2SLC6A4SLC6A3CCNA2
Hydrochloric Acid SCHEMBL9785692 0.69 SLC6A4 (0.63) OPRM1OPRD1OPRK1CHRM3SLC6A2
Trifluoroacetic Acid SCHEMBL21222891 0.69 OPRM1 (0.47) OPRM1OPRD1OPRK1CHRM3SLC6A2
SCHEMBL14882112 0.69 CHRM3 (0.51) CHRM3CYP3A4
SCHEMBL8274719 0.68 CHRM3 (0.36) CHRM3SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL28759723 0.68 CHRNB2 (0.41) SLC6A2SLC6A4SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7491735-B2 Chemokine receptor binding compounds GENZYME CORPORATION (US) 2009-02-17 US disclosed
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
US-20050277670-A1 Chemokine receptor binding compounds ANORMED INC. 2005-12-15 US disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050277670-A1 Chemokine receptor binding compounds CCR5, CXCR3, CCL5 OPRM1 183/4885OPRD1 245/4885OPRK1 158/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.