SCHEMBL426945

SCHEMBL426945

COc1cccc(B2OC(C)(C)C(C)(C)O2)n1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LPL P06858 7/20 0.36
LIPG Q9Y5X9 7/20 0.36
SNCA P37840 1/20 0.34
BTK Q06187 1/20 0.33
EGFR P00533 1/20 0.33
IDH1 O75874 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
DGAT1 O75907 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
ALPL P05186 1/20 0.31
ALOX5 P09917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29699639 1.00 LPL (0.36) LPLLIPGSNCABTKEGFR
SCHEMBL12615775 0.82 LPL (0.33) LPLLIPG
SCHEMBL26653581 0.81 LPL (0.33) LPLLIPG
SCHEMBL31149580 0.80 SNCA (0.38) LPLLIPGSNCADGAT1
SCHEMBL18342256 0.79 LPL (0.39) LPLLIPGIRAK4
SCHEMBL31631018 0.79 LPL (0.39) LPLLIPGIRAK4
SCHEMBL4211647 0.78 LPL (0.40) LPLLIPGDGAT1IRAK4CA1
SCHEMBL31580881 0.77 DGAT1 (0.47) LPLLIPGDGAT1
SCHEMBL1403776 0.77 BRD4 (0.36) LPLLIPG
SCHEMBL17268323 0.77 CCR1 (0.45) LPLLIPGIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 174 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12637427-B2 ALDH-2 inhibitor compounds and methods of use AMYGDALA NEUROSCIENCES, INC. (US) 2026-05-26 US disclosed
US-12590106-B2 Spiromacrocyclic orexin 2 receptor agonists H. LUNDBECK A/S (DK) 2026-03-31 US disclosed
US-12570671-B2 Substituted oxoisoindoline compounds for the treatment of cancer BRISTOL-MYERS SQUIBB COMPANY (US) 2026-03-10 US disclosed
EP-4126843-B1 SUBSTITUTED OXOISOINDOLINE COMPOUNDS FOR THE TREATMENT OF CANCER BRISTOL MYERS SQUIBB CO (US) 2026-02-11 EP disclosed
US-20250263422-A1 SPIROMACROCYCLIC OREXIN 2 RECEPTOR AGONISTS H. LUNDBECK A/S (DK) 2025-08-21 US disclosed
US-20250214970-A1 PYRIDINYLACETAMIDE DERIVATIVES AS SODIUM CHANNEL ACTIVATORS XENON PHARMACEUTICALS INC. (CA) 2025-07-03 US disclosed
EP-4540228-A1 ALDH-2 INHIBITOR COMPOUNDS AND METHODS OF USE Amygdala Neurosciences, Inc. (US) 2025-04-23 EP disclosed
US-20250059185-A1 BICYCLIC HETEROCYCLIC COMPOUNDS USEFUL AS MONOACYLGLYCEROL LIPASE INHIBITORS HOFFMANN-LA ROCHE INC. (US) 2025-02-20 US disclosed
US-20240425521-A1 SPIROMACROCYCLIC OREXIN 2 RECEPTOR AGONISTS H. LUNDBECK A/S (DK) 2024-12-26 US disclosed
EP-4448522-A1 BICYCLIC HETEROCYCLIC COMPOUNDS USEFUL AS MONOACYLGLYCEROL LIPASE INHIBITORS F. Hoffmann-La Roche AG (CH) 2024-10-23 EP disclosed
US-20100190763-A1 Poly (ADP-Ribose) Polymerase (PARP) Inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-07-29 US disclosed
WO-2010085570-A1 Poly (ADP-Ribose) Polymerase (PARP) Inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-07-29 WO disclosed
US-20090305998-A1 HSP90 INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-12-10 US disclosed
US-20090305998-A1 HSP90 INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-12-10 US disclosed
US-20090305998-A1 HSP90 INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-12-10 US disclosed
WO-2009097578-A1 OXIM DERIVATIVES AS HSP90 INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-08-06 WO disclosed
WO-2009097578-A1 OXIM DERIVATIVES AS HSP90 INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-08-06 WO disclosed
US-20080161269-A1 Compounds 620 ASTRAZENECA AB (SE) 2008-07-03 US disclosed
WO-2008076045-A1 NOVEL 2-AMINO- 5-ARYL-IMIDAZOL-4 -ONES ASTRAZENECA AB (SE) 2008-06-26 WO disclosed
WO-2008074997-A1 PYRIDINE BENZAMIDES AND PYRAZINE BENZAMIDES USED AS PKD INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2008-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161269-A1 Compounds 620 MAPT, PSEN1, PSEN2 LPL 3742/4885LIPG 3896/4885SNCA 33/4885
US-20100190763-A1 Poly (ADP-Ribose) Polymerase (PARP) Inhibitors PARP1, PARP3, PARP2 LPL 2097/4885LIPG 2029/4885SNCA 2631/4885
US-20090305998-A1 HSP90 INHIBITORS HSP90AB1, HSP90AA1, HSP90B1 LPL 3355/4885LIPG 3428/4885SNCA 3332/4885
US-20250059185-A1 BICYCLIC HETEROCYCLIC COMPOUNDS USEFUL AS MONOACYLGLYCEROL LIPASE INHIBITORS MGLL, LIPC, PNLIP LPL 5/4885LIPG 14/4885SNCA 4028/4885
US-12570671-B2 Substituted oxoisoindoline compounds for the treatment of cancer NR3C1, NR2C2, RIOX2 LPL 4428/4885LIPG 4384/4885SNCA 4334/4885
US-12590106-B2 Spiromacrocyclic orexin 2 receptor agonists HCRTR2, HCRTR1, OXER1 LPL 4553/4885LIPG 4598/4885SNCA 2821/4885
US-20250214970-A1 PYRIDINYLACETAMIDE DERIVATIVES AS SODIUM CHANNEL ACTIVATORS SCN1A, SCN3A, SCN2A LPL 4564/4885LIPG 4736/4885SNCA 424/4885
US-12637427-B2 ALDH-2 inhibitor compounds and methods of use ALDH3A1, ALDH1A1, ALDH1A2 LPL 188/4885LIPG 2359/4885SNCA 1746/4885
US-20250263422-A1 SPIROMACROCYCLIC OREXIN 2 RECEPTOR AGONISTS HCRTR2, HCRTR1, CRHR2 LPL 4053/4885LIPG 4524/4885SNCA 3068/4885
US-20240425521-A1 SPIROMACROCYCLIC OREXIN 2 RECEPTOR AGONISTS HCRTR2, HCRTR1, CRHR2 LPL 4053/4885LIPG 4524/4885SNCA 3068/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.