Citric Acid

Citric Acid

SCHEMBL428394

CC(O)CO.O=C(O)CC(O)(CC(=O)O)C(=O)O.O=C(O)CC(O)(CC(=O)O)C(=O)O

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACVR1ADORA1ADORA2AADORA2BADORA3ESR1ESR2FLT3GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSC1HRH1HTR7IDH1IDH2IRAK1JAK1JAK2JAK3MEN1OPRM1P2RX3PDE5ASCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASIGMAR1SLC6A2SYKTACR1TOP2ATYK2

The experimentally established mechanism targets of Citric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 1/20 0.37
ALDH1A1 P00352 2/20 0.65
TDP1 Q9NUW8 1/20 0.43
KDM4E B2RXH2 3/20 0.42
TSHR P16473 2/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 2/20 0.42
ALOX15 P16050 1/20 0.42
CPT2 P23786 1/20 0.42
ACLY P53396 1/20 0.42
HMGCR P04035 1/20 0.41
CHRM1 P11229 1/20 0.41
TBXA2R P21731 1/20 0.41
ADRA1A P35348 1/20 0.41
CYP2D6 P10635 2/20 0.39
CYP2C19 P33261 1/20 0.39
HIF1A Q16665 1/20 0.39
SLC13A5 Q86YT5 4/20 0.38
CYP1A2 P05177 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Citric Acid SCHEMBL11971644 1.00 ALDH1A1 (0.65) ALDH1A1TDP1KDM4ETSHRMAPT
Citric Acid SCHEMBL489814 1.00 ALDH1A1 (0.65) ALDH1A1TDP1KDM4ETSHRMAPT
Citric Acid SCHEMBL8626229 1.00 ALDH1A1 (0.65) ALDH1A1TDP1KDM4ETSHRMAPT
Citric Acid SCHEMBL21874899 0.96 ALDH1A1 (0.60) ALDH1A1TDP1KDM4ETSHRMAPT
Citric Acid SCHEMBL1498084 0.89 ALDH1A1 (0.68) ALDH1A1KDM4ETSHRMAPTLMNA
Citric Acid SCHEMBL536573 0.89 ALDH1A1 (0.68) ALDH1A1KDM4ETSHRMAPTLMNA
Citric Acid SCHEMBL28560793 0.89 ALDH1A1 (0.75) ALDH1A1KDM4ETSHRMAPTLMNA
Citric Acid SCHEMBL2199115 0.89 ALDH1A1 (0.75) ALDH1A1KDM4ETSHRMAPTLMNA
Citric Acid SCHEMBL425247 0.87 ALDH1A1 (0.65) ALDH1A1KDM4ETSHRMAPTLMNA
Citric Acid SCHEMBL426131 0.86 ALDH1A1 (0.71) ALDH1A1KDM4ETSHRMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180207085-A1 COSMETIC COMPOSITION BAKEL SRL (IT) 2018-07-26 US claimed
EP-3322488-A1 COSMETIC COMPOSITION Bakel S.R.L. (IT) 2018-05-23 EP claimed
EP-2705828-B1 Quick-penetrating, soft skin care cream DEB IP LTD (GB) 2018-02-14 EP claimed
US-20150231058-A1 QUICK-PENETRATING SOFT SKIN-CARE CREAM EVONIK INDUSTRIES AG (DE) 2015-08-20 US claimed
US-20120020906-A1 ANTIPERSPIRANT SPRAYS WITH ESTER OILS HENKEL AG & CO. KGAA (DE) 2012-01-26 US claimed
EP-3952822-A1 COMPOSITION FOR A TOPICAL APPLICATION ON THE SKIN Biodermic Health & Beauty GmbH & Co. KG (DE) 2022-02-16 EP disclosed
CN-113766906-A Cosmetic composition in the form of a soft solid comprising a hydrophobic powder selected from silica aerogel and polylactic acid, starch and a UV filter system 欧莱雅 2021-12-07 CN disclosed
EP-3853334-A1 POLYSILOXANE-CONTAINING CONCENTRATES WITH IMPROVED STORAGE STABILITY AND USE THEREOF PREFERABLY IN TEXTILE CARE COMPOSITIONS Evonik Operations GmbH (DE) 2021-07-28 EP disclosed
US-11013681-B2 Cosmetic composition BAKEL SRL (IT) 2021-05-25 US disclosed
WO-2020208253-A1 COMPOSITION FOR A TOPICAL APPLICATION ON THE SKIN BIODERMIC HEALTH & BEAUTY GMBH & CO. KG (DE) 2020-10-15 WO disclosed
US-20200138690-A1 COSMETIC COMPOSITIONS COMPRISING AN ASSOCIATIVE POLYURETHANE AND A HYDROPHOBIC COATED PIGMENT L'OREAL (FR) 2020-05-07 US disclosed
EP-3600228-A1 METHOD AND PRODUCT FOR PRODUCING FORMULATIONS CONTAINING CERAMIDE Evonik Operations GmbH (DE) 2020-02-05 EP disclosed
EP-3322488-A1 COSMETIC COMPOSITION Bakel S.R.L. (IT) 2018-05-23 EP disclosed
US-20170157025-A1 TEXTILE FRIENDLY ANTIPERSPIRANT COMPOSITIONS HENKEL AG & CO. KGAA (DE) 2017-06-08 US disclosed
US-20150231058-A1 QUICK-PENETRATING SOFT SKIN-CARE CREAM EVONIK INDUSTRIES AG (DE) 2015-08-20 US disclosed
US-8828367-B2 Water-free antiperspirant non-aerosols in which active substances are more readily released HENKEL AG & CO. KGAA (DE) 2014-09-09 US disclosed
US-8603445-B2 Water-free antiperspirant sprays in which active substances are more readily released HENKEL AG & CO. KGAA (DE) 2013-12-10 US disclosed
US-20120177589-A1 WATER-FREE ANTIPERSPIRANT NON-AEROSOLS IN WHICH ACTIVE SUBSTANCES ARE MORE READILY RELEASED HENKEL AG & CO. KGAA (DE) 2012-07-12 US disclosed
US-20120171143-A1 WATER-FREE ANTIPERSPIRANT SPRAYS IN WHICH ACTIVE SUBSTANCES ARE MORE READILY RELEASED HENKEL AG & CO. KGAA (DE) 2012-07-05 US disclosed
US-20120020906-A1 ANTIPERSPIRANT SPRAYS WITH ESTER OILS HENKEL AG & CO. KGAA (DE) 2012-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120020906-A1 ANTIPERSPIRANT SPRAYS WITH ESTER OILS CUTA, NAPEPLD, LIPE MEN1 2309/4885ALDH1A1 1032/4885TDP1 1145/4885
US-20200138690-A1 COSMETIC COMPOSITIONS COMPRISING AN ASSOCIATIVE POLYURETHANE AND A HYDROPHOBIC COATED PIGMENT MC1R, MCHR1, NACA MEN1 2348/4885ALDH1A1 1667/4885TDP1 1822/4885
US-20120177589-A1 WATER-FREE ANTIPERSPIRANT NON-AEROSOLS IN WHICH ACTIVE SUBSTANCES ARE MORE READILY RELEASED SIGMAR1, POLR1C, CUTA MEN1 4381/4885ALDH1A1 2601/4885TDP1 481/4885
US-20120171143-A1 WATER-FREE ANTIPERSPIRANT SPRAYS IN WHICH ACTIVE SUBSTANCES ARE MORE READILY RELEASED POLR1C, CUTA, PHOSPHO1 MEN1 2543/4885ALDH1A1 1827/4885TDP1 582/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.