SCHEMBL4299065

SCHEMBL4299065

CCN(C)c1ccc(C#N)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.50
ALDH1A1 P00352 3/20 0.44
ADRA2A P08913 2/20 0.44
ADRA2B P18089 2/20 0.44
ADRA2C P18825 2/20 0.44
LOXL2 Q9Y4K0 2/20 0.42
KDM4E B2RXH2 2/20 0.40
GAA P10253 2/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
CA12 O43570 1/20 0.39
CA2 P00918 1/20 0.39
CA3 P07451 1/20 0.39
CA6 P23280 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
MLYCD O95822 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11671854 0.94 TSHR (0.46) CYP2A6ALDH1A1ADRA2AADRA2BADRA2C
SCHEMBL13618783 0.84 CYP2A6 (0.46) CYP2A6ALDH1A1LOXL2KDM4EGAA
SCHEMBL12991122 0.83 MAOA (0.49) ALDH1A1KDM4EGAAMEN1MAPT
SCHEMBL12733256 0.83 CYP2A6 (0.47) CYP2A6ALDH1A1LOXL2MAPTHPGD
SCHEMBL30239355 0.83 DRD2 (0.44) CYP2A6ALDH1A1LOXL2KDM4EGAA
SCHEMBL9174261 0.81 CYP2A6 (0.43) CYP2A6ALDH1A1LOXL2KDM4EGAA
SCHEMBL10330355 0.81 ADRA2A (0.58) CYP2A6ALDH1A1ADRA2AADRA2BADRA2C
SCHEMBL23573064 0.80 CYP2A6 (0.52) CYP2A6ALDH1A1LOXL2KDM4EGAA
SCHEMBL63804 0.80 ALDH1A1 (0.52) CYP2A6ALDH1A1LOXL2KDM4EGAA
SCHEMBL12806211 0.79 HRH3 (0.44) CYP2A6ALDH1A1LOXL2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119431186-A Preparation method of N-alkylamino substituted benzonitrile compound 江苏省农药研究所股份有限公司 2025-02-14 CN disclosed
CN-118290303-A Process for preparing N-methyl-N-substituted-4-cyanoaniline compound 江苏省农药研究所股份有限公司 2024-07-05 CN disclosed
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018113624-A1 FUSED IMIDAZOLE COMPOUND HAVING INDOLEAMINE 2,3-DIOXYGENASE INHIBITORY ACTIVITY 深圳微芯生物科技有限责任公司 2018-06-28 WO disclosed
US-9295673-B2 Combination of mTOR inhibitors and P13-kinase inhibitors, and uses thereof INTELLIKINE LLC (US) 2016-03-29 US disclosed
US-20150320727-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, LLC 2015-11-12 US disclosed
US-20150239894-A1 Amino Compounds for Treatment of Complement Mediated Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2015-08-27 US disclosed
US-20150158859-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE LLC (US) 2015-06-11 US disclosed
US-20150105385-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2015-04-16 US disclosed
US-20150087627-A1 COMBINATION OF KINASE INHIBITORS AND USES THEREOF INTELLIKINE LLC (US) 2015-03-26 US disclosed
US-20120294930-A1 COMBINATION OF KINASE INHIBITORS AND USES THEREOF INTELLIKINE LLC (US) 2012-11-22 US disclosed
WO-2012116237-A2 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, LLC (US) 2012-08-30 WO disclosed
US-20120122838-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. 2012-05-17 US disclosed
US-7851074-B2 Organic electroluminescent display device and chemical compounds for liquid crystals TOHOKU PIONEER CORPORATION (JP) 2010-12-14 US disclosed
US-20090270363-A1 2-Aryl- and 2-Heteroarylthiazolyl Compounds, Methods for Their Preparation and Use Thereof WYETH (US) 2009-10-29 US disclosed
US-20090270363-A1 2-Aryl- and 2-Heteroarylthiazolyl Compounds, Methods for Their Preparation and Use Thereof WYETH (US) 2009-10-29 US disclosed
US-20090270363-A1 2-Aryl- and 2-Heteroarylthiazolyl Compounds, Methods for Their Preparation and Use Thereof WYETH (US) 2009-10-29 US disclosed
WO-2009120826-A1 2-ARYL- AND 2-HETEROARYLTHIAZOLYL COMPOUNDS, METHODS FOR THEIR PREPARATION AND USE THEREOF WYETH (US) 2009-10-01 WO disclosed
US-20090058277-A1 Organic Electroluminescent Display Device and Chemical Compounds for Liquid Crystals TOHOKU PIONEER CORPORATION (JP) 2009-03-05 US disclosed
US-4011173-A MODIFIED NEMATIC MIXTURES WITH POSITIVE DIELECTRIC ANISOTROPY MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-03-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150105385-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PIK3CA, PIK3CD, PIK3CB CYP2A6 2986/4885ALDH1A1 3154/4885ADRA2A 2968/4885
US-20120122838-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PIK3CA, PIK3CD, PIK3CB CYP2A6 2986/4885ALDH1A1 3154/4885ADRA2A 2968/4885
US-20150158859-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PIK3CA, PIK3CD, PIK3CB CYP2A6 2417/4885ALDH1A1 2379/4885ADRA2A 3869/4885
US-20150239894-A1 Amino Compounds for Treatment of Complement Mediated Disorders CFD, TFPI, C9 CYP2A6 4823/4885ALDH1A1 3450/4885ADRA2A 3346/4885
US-20150087627-A1 COMBINATION OF KINASE INHIBITORS AND USES THEREOF MTOR, PIK3CA, AKT1 CYP2A6 4533/4885ALDH1A1 4423/4885ADRA2A 4168/4885
US-20150320727-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PIK3CA, PIK3CD, PIK3CB CYP2A6 2417/4885ALDH1A1 2379/4885ADRA2A 3869/4885
US-20090270363-A1 2-Aryl- and 2-Heteroarylthiazolyl Compounds, Methods for Their Preparation and Use Thereof SEC63, SEC62, SEC22B CYP2A6 1608/4885ALDH1A1 2705/4885ADRA2A 4434/4885
US-20120294930-A1 COMBINATION OF KINASE INHIBITORS AND USES THEREOF MTOR, AKT2, MTMR1 CYP2A6 4607/4885ALDH1A1 4563/4885ADRA2A 4286/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.