SCHEMBL432937

SCHEMBL432937

N#Cc1cccc(C2(C(=O)NCC(c3ccccc3)N3CCCC3)CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
P2RX7 Q99572 3/20 0.42
OPRM1 P35372 1/20 0.41
OPRK1 P41145 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
ELOVL1 Q9BW60 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CNR2 P34972 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL433923 0.85 HSD11B1 (0.49) LMNAP2RX7ALDH1A1MAPTKDM4E
SCHEMBL433444 0.83 SLC6A4 (0.47) LMNASLC6A4P2RX7OPRM1OPRK1
SCHEMBL434266 0.82 MAPT (0.53) LMNAP2RX7OPRM1OPRK1ALDH1A1
SCHEMBL433922 0.82 SMN1; SMN2 (0.53) LMNAP2RX7ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL433170 0.81 SMN1; SMN2 (0.52) LMNAP2RX7ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL433028 0.80 P2RX7 (0.42) LMNAP2RX7ALDH1A1MAPTKDM4E
SCHEMBL432562 0.80 NOS3 (0.40) LMNAP2RX7MAPTKDM4EMEN1
SCHEMBL433030 0.80 SLC6A3 (0.45) P2RX7OPRM1OPRK1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL435636 0.79 HTT (0.48) P2RX7ALDH1A1MAPTKDM4EMEN1
SCHEMBL433860 0.79 P2RX7 (0.55) LMNAP2RX7CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed