SCHEMBL433444

SCHEMBL433444

NC(=O)c1cccc(C2(C(=O)NCC(c3ccccc3)N3CCCC3)CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.47
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
HPGD P15428 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP2C19 P33261 1/20 0.45
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
MAPT P10636 2/20 0.43
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
P2RX7 Q99572 2/20 0.41
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
TP53 P04637 3/20 0.41
LMNA P02545 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL432970 0.89 CYP1A2 (0.44) CYP1A2CYP2C9HPGDMAPK1CYP2C19
Hydrochloric Acid SCHEMBL433923 0.86 HSD11B1 (0.49) CYP1A2CYP2C9HPGDMAPK1CYP2C19
SCHEMBL432937 0.83 LMNA (0.44) SLC6A4CYP1A2CYP2C9HPGDMAPK1
SCHEMBL434266 0.83 MAPT (0.53) CYP1A2CYP2C19MEN1KMT2AMAPT
SCHEMBL433922 0.82 SMN1; SMN2 (0.53) CYP1A2CYP2C9HPGDMAPK1CYP2C19
Hydrochloric Acid SCHEMBL433170 0.82 SMN1; SMN2 (0.52) CYP1A2CYP2C9HPGDMAPK1CYP2C19
Hydrochloric Acid SCHEMBL433028 0.81 P2RX7 (0.42) MEN1KMT2AMAPTP2RX7ROCK2
SCHEMBL433833 0.81 OPRM1 (0.47) MEN1KMT2AMAPTOPRM1OPRD1
SCHEMBL433030 0.81 SLC6A3 (0.45) MEN1KMT2AMAPTOPRM1OPRK1
Hydrochloric Acid SCHEMBL435636 0.80 HTT (0.48) MEN1KMT2AMAPTP2RX7L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed