SCHEMBL434266

SCHEMBL434266

COc1cccc(C2(C(=O)NCC(c3ccccc3)N3CCCC3)CC2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.53
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 1/20 0.53
P2RX7 Q99572 3/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
RAB9A P51151 1/20 0.50
PKM P14618 1/20 0.49
OPRM1 P35372 1/20 0.49
OPRD1 P41143 1/20 0.49
OPRK1 P41145 1/20 0.49
OPRL1 P41146 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
HSD17B10 Q99714 1/20 0.49
LMNA P02545 2/20 0.48
TP53 P04637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL435915 0.89 P2RX7 (0.60) MAPTKDM4EALDH1A1P2RX7MEN1
Hydrochloric Acid SCHEMBL435636 0.87 HTT (0.48) MAPTKDM4EALDH1A1P2RX7MEN1
Hydrochloric Acid SCHEMBL433923 0.85 HSD11B1 (0.49) MAPTKDM4EALDH1A1P2RX7MEN1
SCHEMBL433444 0.83 SLC6A4 (0.47) MAPTKDM4EALDH1A1P2RX7MEN1
Hydrochloric Acid SCHEMBL433028 0.82 P2RX7 (0.42) MAPTKDM4EALDH1A1P2RX7MEN1
SCHEMBL432937 0.82 LMNA (0.44) MAPTKDM4EALDH1A1P2RX7MEN1
SCHEMBL433922 0.82 SMN1; SMN2 (0.53) ALDH1A1P2RX7MEN1KMT2AL3MBTL1
SCHEMBL433030 0.82 SLC6A3 (0.45) MAPTKDM4EALDH1A1P2RX7MEN1
Hydrochloric Acid SCHEMBL433170 0.81 SMN1; SMN2 (0.52) ALDH1A1P2RX7MEN1KMT2AL3MBTL1
SCHEMBL433833 0.80 OPRM1 (0.47) MAPTKDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed