SCHEMBL433030

SCHEMBL433030

CS(=O)(=O)Nc1cccc(C2(C(=O)NCC(c3ccccc3)N3CCCC3)CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 2/20 0.45
UBE2N P61088 1/20 0.43
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
OPRM1 P35372 1/20 0.40
PRMT5 O14744 1/20 0.40
P2RX7 Q99572 2/20 0.39
OPRK1 P41145 1/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL433028 0.86 P2RX7 (0.42) MAPTKDM4EALDH1A1P2RX7ROCK2
SCHEMBL433833 0.85 OPRM1 (0.47) MAPTKDM4EALDH1A1OPRM1OPRK1
SCHEMBL435352 0.84 P2RX7 (0.43) SLC6A3MAPTKDM4EALDH1A1P2RX7
Hydrochloric Acid SCHEMBL433923 0.82 HSD11B1 (0.49) MAPTKDM4EALDH1A1P2RX7MEN1
SCHEMBL435241 0.82 P2RX7 (0.42) SLC6A3MAPTKDM4EALDH1A1P2RX7
SCHEMBL434266 0.82 MAPT (0.53) MAPTKDM4EALDH1A1OPRM1P2RX7
SCHEMBL435467 0.81 ALDH1A1 (0.44) MAPTKDM4EALDH1A1P2RX7MEN1
SCHEMBL434790 0.81 OPRM1 (0.47) KDM4EALDH1A1OPRM1P2RX7OPRK1
SCHEMBL433444 0.81 SLC6A4 (0.47) MAPTKDM4EALDH1A1OPRM1P2RX7
SCHEMBL432937 0.80 LMNA (0.44) MAPTKDM4EALDH1A1OPRM1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO claimed
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed