SCHEMBL433860

SCHEMBL433860

O=C(NCC(c1ccccc1)N1CCCC1)C1(c2ccc(Cl)cc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.55
TRPA1 O75762 7/20 0.54
TP53 P04637 4/20 0.54
CYP3A4 P08684 1/20 0.52
CYP2C8 P10632 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
KCNH2 Q12809 1/20 0.52
LMNA P02545 2/20 0.51
HSD11B1 P28845 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL433923 0.91 HSD11B1 (0.49) P2RX7TP53CYP2C9CYP2C19LMNA
SCHEMBL433922 0.87 SMN1; SMN2 (0.53) P2RX7TRPA1TP53CYP2C9CYP2C19
SCHEMBL432970 0.87 CYP1A2 (0.44) P2RX7TRPA1TP53CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL433170 0.86 SMN1; SMN2 (0.52) P2RX7TRPA1TP53CYP2C9CYP2C19
SCHEMBL435915 0.86 P2RX7 (0.60) P2RX7TP53LMNA
SCHEMBL435467 0.85 ALDH1A1 (0.44) P2RX7TRPA1TP53CYP2C9CYP2C19
SCHEMBL434779 0.84 POLB (0.52) P2RX7TP53CYP2D6LMNA
SCHEMBL434790 0.82 OPRM1 (0.47) P2RX7TRPA1CYP2D6
SCHEMBL434036 0.81 TP53 (0.54) TP53LMNA
SCHEMBL4963409 0.81 TRPA1 (0.52) TRPA1CYP3A4CYP2C8CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed