SCHEMBL4396992

SCHEMBL4396992

COc1ccc(-c2cccc3[nH]c(OC(=O)NC4CCN(CCN5CCCCCC5)CC4)cc23)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
SIGMAR1 Q99720 2/20 0.40
MCHR1 Q99705 2/20 0.40
MEN1 O00255 1/20 0.40
CCR5 P51681 1/20 0.40
CHRM3 P20309 1/20 0.40
HTR4 Q13639 1/20 0.39
DRD4 P21917 1/20 0.39
KCNH2 Q12809 1/20 0.39
DYRK1A Q13627 1/20 0.38
KDM4E B2RXH2 1/20 0.38
FAAH O00519 2/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
ACKR3 P25106 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4551165 0.93 SIGMAR1 (0.40) KMT2ASIGMAR1MCHR1CCR5CHRM3
SCHEMBL4396457 0.92 HRH3 (0.42) KMT2AKCNH2KDM4EFAAH
SCHEMBL4410349 0.92 HRH3 (0.42) KMT2AKCNH2KDM4EFAAH
SCHEMBL4396410 0.91 L3MBTL1 (0.40) MCHR1DYRK1AKDM4EFAAH
SCHEMBL4396337 0.90 HTR7 (0.43) KMT2AMEN1KDM4EFAAH
SCHEMBL4405570 0.90 TLR7 (0.43) KMT2ASIGMAR1HTR4DYRK1AKDM4E
SCHEMBL4405673 0.89 CHRM3 (0.42) MCHR1CHRM3DRD4KCNH2DYRK1A
SCHEMBL4406646 0.89 TSHR (0.42) KMT2ASIGMAR1MCHR1MEN1HTR4
SCHEMBL4394199 0.89 CHRM3 (0.41) CHRM3HTR4DYRK1AFAAHACKR3
SCHEMBL4396957 0.89 TLR9 (0.42) SIGMAR1HTR4DYRK1AACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed