SCHEMBL4485668

SCHEMBL4485668

CC(Cc1ccccc1)c1c(-c2ccncc2)[nH]c(C=O)c1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
CYP3A4 P08684 1/20 0.39
CDC7 O00311 2/20 0.37
ROCK2 O75116 3/20 0.36
ROCK1 Q13464 3/20 0.36
RPS6KA5 O75582 1/20 0.36
RPS6KA4 O75676 1/20 0.36
PRKACA P17612 1/20 0.36
MAPK1 P28482 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
IRAK1 P51617 1/20 0.36
PRKX P51817 1/20 0.36
PRKG1 Q13976 1/20 0.36
PKN2 Q16513 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
SGK2 Q9HBY8 1/20 0.36
FNTA P49354 4/20 0.36
FNTB P49356 4/20 0.36
BRAF P15056 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4494581 0.92 ESR1 (0.38) ALDH1A1CNR1
SCHEMBL4490045 0.85 PPARG (0.42) ALDH1A1
SCHEMBL4498684 0.83 CSNK1D (0.44) CDC7GSK3BCSNK1A1CSNK1DCLK2
SCHEMBL4504906 0.83 MEN1 (0.45) ALDH1A1MAPK1CNR1
SCHEMBL4559834 0.83 PPARG (0.41) ALDH1A1
SCHEMBL4492334 0.81 TAAR1 (0.36)
SCHEMBL4504872 0.81 LDHA (0.38) FNTAFNTB
SCHEMBL4485738 0.80 MTNR1A (0.41) ALDH1A1
SCHEMBL4477477 0.79 TDP1 (0.42) ALDH1A1
SCHEMBL4481909 0.78 KDM4E (0.40) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed