SCHEMBL4492334

SCHEMBL4492334

CC(Cc1ccccc1)c1c(I)[nH]c(C=O)c1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ALOX5 P09917 2/20 0.34
LDHA P00338 1/20 0.34
LDHB P07195 1/20 0.34
CYP1A2 P05177 1/20 0.34
CTRB1 P17538 3/20 0.33
LMNA P02545 1/20 0.33
ALB P02768 1/20 0.33
ESR1 P03372 1/20 0.33
RARB P10826 1/20 0.33
CYP2C9 P11712 1/20 0.33
ADRB3 P13945 1/20 0.33
NFKB1 P19838 1/20 0.33
PTGS1 P23219 1/20 0.33
HTR2A P28223 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4494581 0.86 ESR1 (0.38) TAAR1MEN1KMT2ANPC1RAB9A
SCHEMBL4485668 0.81 ALDH1A1 (0.39)
SCHEMBL4504872 0.80 LDHA (0.38) TAAR1MEN1KMT2ANPC1RAB9A
SCHEMBL4490045 0.79 PPARG (0.42) MEN1KMT2ARAB9ALDHACYP1A2
SCHEMBL4504906 0.78 MEN1 (0.45) MEN1KMT2ANPC1RAB9A
SCHEMBL4481909 0.77 KDM4E (0.40) TAAR1MEN1KMT2ANPC1RAB9A
SCHEMBL4559834 0.77 PPARG (0.41) MEN1KMT2ANPC1RAB9AALOX5
SCHEMBL4485206 0.77 ALDH1A1 (0.32) TAAR1MEN1KMT2ANPC1RAB9A
SCHEMBL4491379 0.65 FBP1 (0.34) KMT2ALDHALDHB
SCHEMBL4492326 0.65 RAB9A (0.51) MEN1KMT2ANPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed