SCHEMBL4491745

SCHEMBL4491745

CCc1c(C(=O)O)c(C=O)n(C)c1-c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AR P10275 8/20 0.43
TSPO P30536 1/20 0.42
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 3/20 0.37
RAB9A P51151 2/20 0.36
PKM P14618 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
MAPK1 P28482 1/20 0.36
HRH2 P25021 1/20 0.36
HRH1 P35367 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4491009 0.83 ALDH1A1 (0.43) ALDH1A1RAB9AKDM4EPOLBMAPT
SCHEMBL4490745 0.82 GRIA2 (0.40) ALDH1A1KDM4EMAPK1
SCHEMBL4504902 0.82 AR (0.57) ARALDH1A1KDM4EPOLBMAPT
SCHEMBL4498679 0.80 CCNC (0.36) ALDH1A1RAB9AKDM4EPOLBMAPT
SCHEMBL4495477 0.78 ALDH1A1 (0.42) ARTDP1ALDH1A1RAB9AKDM4E
SCHEMBL4477472 0.71 PGR (0.48) ARALDH1A1KDM4EMAPT
SCHEMBL4480912 0.68
SCHEMBL4496740 0.68 GRM5 (0.39) RAB9AKDM4EPOLBMAPT
SCHEMBL4500631 0.68 DHODH (0.37) ARALDH1A1PKMKDM4E
SCHEMBL4504195 0.68 CCR1 (0.38) ALDH1A1RAB9APKMKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed