SCHEMBL4477472

SCHEMBL4477472

CCc1c(C(=O)O)c(C=O)n(Cc2ccccc2)c1-c1cccc([N+](=O)[O-])c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PGR P06401 2/20 0.48
ALDH1A1 P00352 2/20 0.48
GAA P10253 2/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
HPGD P15428 1/20 0.48
AR P10275 3/20 0.47
MAPT P10636 2/20 0.47
CFTR P13569 6/20 0.46
CCR2 P41597 1/20 0.42
CYP19A1 P11511 1/20 0.42
FEN1 P39748 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
PLA2G2A P14555 2/20 0.41
KMT2A Q03164 1/20 0.41
RECQL P46063 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4504902 0.89 AR (0.57) ALDH1A1KDM4ELMNAARMAPT
SCHEMBL4494579 0.85 ALDH1A1 (0.43) ALDH1A1KDM4ELMNAHPGDAR
SCHEMBL4559832 0.84 TP53 (0.46) ALDH1A1GAALMNAHPGDMAPT
SCHEMBL4490747 0.84 PGR (0.43) PGRALDH1A1GAAKDM4ELMNA
SCHEMBL4485732 0.82 KMT2A (0.47) CCR2FEN1PLA2G2AKMT2A
SCHEMBL4484664 0.81 CFTR (0.45) ALDH1A1LMNAARCFTRCCR2
SCHEMBL4485664 0.78 KDM4E (0.40) ALDH1A1KDM4ELMNAMAPTSMN1; SMN2
SCHEMBL4490040 0.76 GFER (0.47) ALDH1A1GAAKDM4EHPGDMAPT
SCHEMBL4492336 0.75 AR (0.47) ALDH1A1GAAKDM4ELMNAHPGD
SCHEMBL4504869 0.74 ALDH1A1 (0.42) ALDH1A1LMNAMAPTSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed