SCHEMBL4540032

SCHEMBL4540032

COc1ccc(S(=O)(=O)N2CCC(CC(=O)NC34CC5CC(CC(C5)C3)C4)C2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.51
EPHX1 P07099 1/20 0.49
MMP9 P14780 2/20 0.48
MMP1 P03956 1/20 0.48
MMP3 P08254 1/20 0.48
MMP7 P09237 1/20 0.48
MMP13 P45452 1/20 0.48
CNR2 P34972 1/20 0.48
ALDH1A1 P00352 2/20 0.47
LMNA P02545 3/20 0.47
GAA P10253 2/20 0.47
EPHX2 P34913 2/20 0.47
NPC1 O15118 1/20 0.46
TSHR P16473 3/20 0.46
HTT P42858 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
ALOX12 P18054 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MAPT P10636 1/20 0.46
MMP2 P08253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4537319 0.95 ALDH1A1 (0.52) PKMEPHX1MMP9MMP1MMP3
SCHEMBL4541877 0.94 PKM (0.56) PKMEPHX1MMP9MMP1MMP3
SCHEMBL4535944 0.89 EPHX1 (0.52) EPHX1ALDH1A1LMNAEPHX2TSHR
SCHEMBL4541355 0.89 USP2 (0.53) PKMEPHX1CNR2ALDH1A1LMNA
SCHEMBL4539274 0.87 CYP3A4 (0.51) PKMEPHX1ALDH1A1LMNAEPHX2
SCHEMBL4536776 0.87 LMNA (0.62) EPHX1ALDH1A1LMNAEPHX2NPC1
SCHEMBL4540431 0.86 NPC1 (0.55) PKMEPHX1ALDH1A1LMNAGAA
SCHEMBL4535739 0.86 EPHX2 (0.54) PKMEPHX1ALDH1A1LMNAEPHX2
SCHEMBL4543052 0.85 NPC1 (0.48) EPHX1CNR2ALDH1A1LMNAEPHX2
SCHEMBL4542516 0.85 LMNA (0.49) EPHX1ALDH1A1LMNAGAAEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed