SCHEMBL4542516

SCHEMBL4542516

O=C(CC1CCN(S(=O)(=O)c2ccc(C(F)(F)F)cc2)C1)NC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.47
EPHX1 P07099 3/20 0.47
TSHR P16473 1/20 0.47
ALOX12 P18054 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
EPHX2 P34913 2/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
TRPV4 Q9HBA0 4/20 0.44
CCR6 P51684 1/20 0.42
CACNA1B Q00975 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4539395 0.95 LMNA (0.47) LMNAALDH1A1GAAEPHX1TSHR
SCHEMBL4540917 0.94 LMNA (0.53) LMNAALDH1A1GAAEPHX1TSHR
SCHEMBL4539274 0.90 CYP3A4 (0.51) LMNAALDH1A1EPHX1TSHRALOX12
SCHEMBL4537706 0.88 EPHX2 (0.48) LMNAGAAEPHX1EPHX2MEN1
SCHEMBL4535944 0.88 EPHX1 (0.52) LMNAALDH1A1EPHX1TSHRALOX12
SCHEMBL4536776 0.88 LMNA (0.62) LMNAALDH1A1EPHX1TSHRALOX12
SCHEMBL4540431 0.87 NPC1 (0.55) LMNAALDH1A1GAAEPHX1TSHR
SCHEMBL4537391 0.87 EPHX1 (0.53) LMNAALDH1A1GAAEPHX1EPHX2
SCHEMBL4543052 0.86 NPC1 (0.48) LMNAALDH1A1EPHX1TSHRALOX12
SCHEMBL4540032 0.85 PKM (0.51) LMNAALDH1A1GAAEPHX1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed