SCHEMBL4551382

SCHEMBL4551382

CCOc1cc(CN(c2ccc(C(F)(F)F)cn2)C2CCNCC2)ccc1OC

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PDE4B Q07343 1/20 0.40
REN P00797 2/20 0.39
SLC6A2 P23975 4/20 0.39
SLC6A4 P31645 4/20 0.39
RAB9A P51151 1/20 0.39
TACR1 P25103 3/20 0.38
HTR2A P28223 3/20 0.38
SLC6A3 Q01959 1/20 0.38
HPGD P15428 1/20 0.36
MAP4K3 Q8IVH8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973911 0.85 SLC6A2 (0.40) PDE4BRENSLC6A2SLC6A4SLC6A3
SCHEMBL3972925 0.83 MAPK1 (0.44) ALDH1A1NPSR1RENSLC6A2SLC6A4
SCHEMBL3973856 0.83 L3MBTL1 (0.47) ALDH1A1NPSR1REN
SCHEMBL3974580 0.83 REN (0.41) KDM4EALDH1A1NPSR1RENSLC6A2
SCHEMBL3977756 0.83 REN (0.41) KDM4EALDH1A1RENTACR1HTR2A
SCHEMBL3973369 0.83 REN (0.43) KDM4EALDH1A1NPSR1RENSLC6A2
SCHEMBL3974286 0.82 REN (0.43) KDM4EALDH1A1NPSR1REN
SCHEMBL3979346 0.79 REN (0.43) ALDH1A1RENSLC6A2SLC6A4SLC6A3
SCHEMBL4551389 0.79 MC4R (0.46) KDM4EALDH1A1RENSLC6A2SLC6A4
SCHEMBL4544203 0.78 SLC6A2 (0.45) KDM4EALDH1A1NPSR1RENSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed