SCHEMBL4551389

SCHEMBL4551389

CCOc1cc(CN(c2ccc3cc(F)ccc3n2)C2CCNCC2)ccc1OC

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.46
SLC6A2 P23975 11/20 0.43
SLC6A4 P31645 10/20 0.43
SLC6A3 Q01959 7/20 0.40
REN P00797 1/20 0.38
HTR1A P08908 1/20 0.37
FGFR1 P11362 1/20 0.35
FGFR2 P21802 1/20 0.35
FGFR4 P22455 1/20 0.35
FGFR3 P22607 1/20 0.35
KDR P35968 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KCNH2 Q12809 1/20 0.35
TACR1 P25103 1/20 0.35
KDM4E B2RXH2 1/20 0.35
APAF1 O14727 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4551382 0.79 KDM4E (0.42) SLC6A2SLC6A4SLC6A3RENTACR1
SCHEMBL4544203 0.78 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3RENMEN1
SCHEMBL3972925 0.78 MAPK1 (0.44) MC4RSLC6A2SLC6A4SLC6A3REN
SCHEMBL3931492 0.77 REN (0.41) MC4RSLC6A2SLC6A4SLC6A3REN
SCHEMBL3973911 0.77 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3REN
SCHEMBL3973856 0.76 L3MBTL1 (0.47) RENMEN1KMT2AALDH1A1MAPT
SCHEMBL3973369 0.75 REN (0.43) SLC6A2SLC6A4SLC6A3RENKCNH2
SCHEMBL3973450 0.74 SLC6A2 (0.52) SLC6A2SLC6A4SLC6A3RENKCNH2
SCHEMBL3974286 0.74 REN (0.43) RENMEN1KMT2AKDM4EALDH1A1
SCHEMBL3974580 0.74 REN (0.41) SLC6A2SLC6A4RENMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed