SCHEMBL4595333

SCHEMBL4595333

C=CCC1CNC(=O)N1CC=C

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.34
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15422827 0.77 ALDH1A1 (0.34) ALDH1A1
SCHEMBL4543295 0.76 CYP3A4 (0.35) CYP3A4MAPTL3MBTL1POLB
SCHEMBL1077227 0.76 CYP3A4 (0.35) CYP3A4MAPTL3MBTL1POLB
SCHEMBL3313650 0.73 CYP3A4 (0.33) CYP3A4
SCHEMBL30479506 0.66 CYP3A4 (0.41) CYP3A4ALDH1A1MAPTL3MBTL1POLB
SCHEMBL5135057 0.66 CYP3A4 (0.41) CYP3A4ALDH1A1MAPTL3MBTL1
SCHEMBL6569507 0.64 P2RX7 (0.30)
SCHEMBL16139578 0.64 P2RX7 (0.32) L3MBTL1
SCHEMBL18106821 0.63 CYP3A4 (0.42) CYP3A4ALDH1A1MAPTL3MBTL1POLB
SCHEMBL24591674 0.62 CYP3A4 (0.46) CYP3A4ALDH1A1MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12551434-B2 Zwitterionic polymer particle compositions and related methods WAYNE STATE UNIVERSITY (US) 2026-02-17 US claimed
US-20230225969-A1 ZWITTERIONIC POLYMER PARTICLE COMPOSITIONS AND RELATED METHODS WAYNE STATE UNIVERSITY 2023-07-20 US claimed
WO-2021236922-A1 ZWITTERIONIC POLYMER PARTICLE COMPOSITIONS AND RELATED METHODS WAYNE STATE UNIVERSITY (US) 2021-11-25 WO claimed
EP-3261626-A1 METHODS AND COMPOSITIONS RELATING TO BIOCOMPATIBLE IMPLANTS Wayne State University (US) 2018-01-03 EP claimed
WO-2016138528-A1 METHODS AND COMPOSITIONS RELATING TO BIOCOMPATIBLE IMPLANTS WAYNE STATE UNIVERSITY (US) 2016-09-01 WO claimed
EP-1572759-B1 PROCESS FOR MAKING A VINYL AMIDE POLYMER COMPOSITION FOR SKIN AND HAIR COMPOSITIONS ISP INVESTMENTS INC (US) 2008-01-02 EP claimed
EP-1572759-A4 PROCESS FOR MAKING A VINYL AMIDE POLYMER COMPOSITION FOR SKIN AND HAIR COMPOSITIONS ISP INVESTMENTS INC (US) 2006-11-08 EP claimed
EP-1037929-B1 NON-AQUEOUS, HETEROGENEOUS POLYMERIZATION PROCESS AND REACTION PRODUCT OBTAINED THEREBY ISP INVESTMENTS INC (US) 2006-07-12 EP claimed
EP-1572759-A1 PROCESS FOR MAKING A VINYL AMIDE POLYMER COMPOSITION FOR SKIN AND HAIR COMPOSITIONS ISP INVESTMENTS INC. (US) 2005-09-14 EP claimed
EP-1037929-A4 NON-AQUEOUS, HETEROGENEOUS POLYMERIZATION PROCESS AND REACTION PRODUCT OBTAINED THEREBY ISP INVESTMENTS INC (US) 2004-09-15 EP claimed
WO-2004046212-A1 PROCESS FOR MAKING A VINYL AMIDE POLYMER COMPOSITION FOR SKIN AND HAIR COMPOSITIONS ISP INVESTMENTS INC. (US) 2004-06-03 WO claimed
US-6566473-B1 Process for making a vinyl amide polymer composition for skin and hair compositions ISP INVESTMENTS INC. 2003-05-20 US claimed
US-6300442-B1 Process for making a cosmetically or pharmaceutically-acceptable emulsion or gel composition ISP INVESTMENTS INC. 2001-10-09 US claimed
EP-0590491-B1 Soluble anionic polymerization initiators and products therefrom BRIDGESTONE CORP (JP) 2001-07-11 EP claimed
US-6255421-B1 Non-aqueous, heterogeneous polymerization process and reaction product obtained thereby ISP INVESTMENTS INC. 2001-07-03 US claimed
EP-1037929-A1 NON-AQUEOUS, HETEROGENEOUS POLYMERIZATION PROCESS AND REACTION PRODUCT OBTAINED THEREBY ISP INVESTMENTS INC. (US) 2000-09-27 EP claimed
US-6048522-A Controlled-release, drug-delivery composition ISP INVESTMENTS INC. (US) 2000-04-11 US claimed
WO-1999029735-A1 NON-AQUEOUS, HETEROGENEOUS POLYMERIZATION PROCESS AND REACTION PRODUCT OBTAINED THEREBY ISP INVESTMENTS INC. (US) 1999-06-17 WO claimed
EP-0590491-A2 Soluble anionic polymerization initiators and products therefrom BRIDGESTONE CORPORATION (JP) 1994-04-06 EP claimed
JP-7233330-A None JP disclosed
US-12551434-B2 Zwitterionic polymer particle compositions and related methods WAYNE STATE UNIVERSITY (US) 2026-02-17 US disclosed
US-12257309-B2 Zwitterionic polymer-insulin compositions and related methods WAYNE STATE UNIVERSITY (US) 2025-03-25 US disclosed
US-20230398265-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF TISSUE ADHESION NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-12-14 US disclosed
US-20230225969-A1 ZWITTERIONIC POLYMER PARTICLE COMPOSITIONS AND RELATED METHODS WAYNE STATE UNIVERSITY 2023-07-20 US disclosed
EP-3570874-B1 ZWITTERIONIC POLYMER-INSULIN COMPOSITIONS AND RELATED METHODS UNIV WAYNE STATE (US) 2023-03-08 EP disclosed
US-11591287-B2 Antifouling zwitterionic polymer coating and reverse coating method WAYNE STATE UNIVERSITY (US) 2023-02-28 US disclosed
WO-2022103768-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF TISSUE ADHESION WAYNE STATE UNIVERSITY (US) 2022-05-19 WO disclosed
US-20220125937-A1 ZWITTERIONIC POLYMER-INSULIN COMPOSITIONS AND RELATED METHODS WAYNE STATE UNIVERSITY 2022-04-28 US disclosed
WO-2022040513-A1 COATING COMPOSITIONS AND METHODS WAYNE STATE UNIVERSITY (US) 2022-02-24 WO disclosed
WO-2021236922-A1 ZWITTERIONIC POLYMER PARTICLE COMPOSITIONS AND RELATED METHODS WAYNE STATE UNIVERSITY (US) 2021-11-25 WO disclosed
US-20200181426-A1 ANTIFOULING ZWITTERIONIC POLYMER COATING AND REVERSE COATING METHOD WAYNE STATE UNIVERSITY (US) 2020-06-11 US disclosed
US-10596300-B2 Methods and compositions relating to biocompatible implants WAYNE STATE UNIVERSITY (US) 2020-03-24 US disclosed
WO-2018226854-A2 ANTIFOULING POLYMER COATINGS AND REVERSE COATING METHOD WAYNE STATE UNIVERSITY (US) 2018-12-13 WO disclosed
US-20180236135-A1 METHODS AND COMPOSITIONS RELATING TO BIOCOMPATIBLE IMPLANTS WAYNE STATE UNIVERSITY 2018-08-23 US disclosed
WO-2018136505-A1 ZWITTERIONIC POLYMER-INSULIN COMPOSITIONS AND RELATED METHODS WAYNE STATE UNIVERSITY (US) 2018-07-26 WO disclosed
EP-3261626-A1 METHODS AND COMPOSITIONS RELATING TO BIOCOMPATIBLE IMPLANTS Wayne State University (US) 2018-01-03 EP disclosed
WO-2016138528-A1 METHODS AND COMPOSITIONS RELATING TO BIOCOMPATIBLE IMPLANTS WAYNE STATE UNIVERSITY (US) 2016-09-01 WO disclosed
US-7371369-B2 Polymeric interpenetrated network carrier and serial polymerization involving a crosslinked polymer network ISP INVESTMENTS INC. (US) 2008-05-13 US disclosed
EP-1572759-B1 PROCESS FOR MAKING A VINYL AMIDE POLYMER COMPOSITION FOR SKIN AND HAIR COMPOSITIONS ISP INVESTMENTS INC (US) 2008-01-02 EP disclosed
EP-1572759-A4 PROCESS FOR MAKING A VINYL AMIDE POLYMER COMPOSITION FOR SKIN AND HAIR COMPOSITIONS ISP INVESTMENTS INC (US) 2006-11-08 EP disclosed
EP-1037929-B1 NON-AQUEOUS, HETEROGENEOUS POLYMERIZATION PROCESS AND REACTION PRODUCT OBTAINED THEREBY ISP INVESTMENTS INC (US) 2006-07-12 EP disclosed
EP-1572759-A1 PROCESS FOR MAKING A VINYL AMIDE POLYMER COMPOSITION FOR SKIN AND HAIR COMPOSITIONS ISP INVESTMENTS INC. (US) 2005-09-14 EP disclosed
WO-2005046582-A2 POLYMERIC INTERPENETRATED NETWORK CARRIER AND SERIAL POLYMERIZATION INVOLVING A CROSSLINKED POLYMER NETWORK ISP INVESTMENTS INC. (US) 2005-05-26 WO disclosed
US-20050101721-A1 Polymeric interpenetrated network carrier and serial polymerization involving a crosslinked polymer network PHARMACHEM LABORATORIES LLC 2005-05-12 US disclosed
EP-1037929-A4 NON-AQUEOUS, HETEROGENEOUS POLYMERIZATION PROCESS AND REACTION PRODUCT OBTAINED THEREBY ISP INVESTMENTS INC (US) 2004-09-15 EP disclosed
WO-2004046212-A1 PROCESS FOR MAKING A VINYL AMIDE POLYMER COMPOSITION FOR SKIN AND HAIR COMPOSITIONS ISP INVESTMENTS INC. (US) 2004-06-03 WO disclosed
US-6566473-B1 Process for making a vinyl amide polymer composition for skin and hair compositions ISP INVESTMENTS INC. 2003-05-20 US disclosed
US-6300442-B1 Process for making a cosmetically or pharmaceutically-acceptable emulsion or gel composition ISP INVESTMENTS INC. 2001-10-09 US disclosed
US-6255421-B1 Non-aqueous, heterogeneous polymerization process and reaction product obtained thereby ISP INVESTMENTS INC. 2001-07-03 US disclosed
US-6177068-B1 Vinyl amide polymer delivery system for hair and skin treating compositions ISP INVESTMENTS INC. 2001-01-23 US disclosed
EP-1037929-A1 NON-AQUEOUS, HETEROGENEOUS POLYMERIZATION PROCESS AND REACTION PRODUCT OBTAINED THEREBY ISP INVESTMENTS INC. (US) 2000-09-27 EP disclosed
US-6048522-A Controlled-release, drug-delivery composition ISP INVESTMENTS INC. (US) 2000-04-11 US disclosed
WO-1999029735-A1 NON-AQUEOUS, HETEROGENEOUS POLYMERIZATION PROCESS AND REACTION PRODUCT OBTAINED THEREBY ISP INVESTMENTS INC. (US) 1999-06-17 WO disclosed
US-5716634-A CONSISTING OF MICROPARTICLES OF SPECIFIED SIZE AND HAVING SPECIFIED VISCOSITY; CARRIER FOR COSMETICS, DRUGS ISP INVESTMENTS INC. (US) 1998-02-10 US disclosed
US-5654385-A One-step process for making lightly-crosslinked polyvinylpyrrolidone hydrogel ISP INVESTMENTS INC. (US) 1997-08-05 US disclosed
US-5614583-A Homogenized flowable hydrogel of crosslinked N-vinyl lactam polymer ISP INVESTMENTS INC. (US) 1997-03-25 US disclosed
WO-1997009965-A1 A NON-IRRITATING SKIN AND HAIR REJUVENATING COMPOSITION HAVING A pH BETWEEN 1 AND 6.5 ISP INVESTMENTS INC. (US) 1997-03-20 WO disclosed
US-5605685-A CROSSLINKED N-VINYL LACTAM HYDROGEL AND ONE OF PYRUVIC ACID, MONO- AND POLYCARBOXYLATED HYDROCARBONS OPTIONALLY SUBSTITUTED WITH HYDROXY, AND AN AMMONIUM OR ALKALI METAL SALT OF THE PRECEDING COMPOUNDS ISP INVESTMENTS INC. (US) 1997-02-25 US disclosed
JP-H07233330-A PRODUCTION OF DIANTHRAQUINONE-N,N'-DIHYDROAZINE MITSUI TOATSU CHEM INC 1995-09-05 JP disclosed
US-5393825-A Films and extrusions of cured crosslinked vinyl lactam polymer and method of preparation ISP INVESTMENTS INC. (US) 1995-02-28 US disclosed
US-5354823-A Films and extrusions of cured crosslinked vinyl lactam polymer and method of preparation ISP INVESTMENTS INC. (US) 1994-10-11 US disclosed
US-5336697-A Molded cellular crosslinked vinyl lactam polymer gel and method of preparation ISP INVESTMENTS INC. (US) 1994-08-09 US disclosed
US-5280049-A Molded cellular crosslinked vinyl lactam polymer gel and method of preparation ISP INVESTMENTS INC. (US) 1994-01-18 US disclosed
US-5280049-A Molded cellular crosslinked vinyl lactam polymer gel and method of preparation ISP INVESTMENTS INC. (US) 1994-01-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230225969-A1 ZWITTERIONIC POLYMER PARTICLE COMPOSITIONS AND RELATED METHODS IAPP, IGFBP6, SI CYP3A4 4582/4885ALDH1A1 4697/4885MAPT 4555/4885
US-11591287-B2 Antifouling zwitterionic polymer coating and reverse coating method ITGA5, GFER, EPCAM CYP3A4 4358/4885ALDH1A1 2445/4885MAPT 1651/4885
US-20180236135-A1 METHODS AND COMPOSITIONS RELATING TO BIOCOMPATIBLE IMPLANTS CD44, ILK, CRYAA CYP3A4 3428/4885ALDH1A1 1067/4885MAPT 4224/4885
US-20230398265-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF TISSUE ADHESION PLOD3, ICAM1, ITGB3 CYP3A4 4058/4885ALDH1A1 352/4885MAPT 3409/4885
US-12257309-B2 Zwitterionic polymer-insulin compositions and related methods IAPP, INSR, IRS1 CYP3A4 4617/4885ALDH1A1 4850/4885MAPT 1304/4885
US-12551434-B2 Zwitterionic polymer particle compositions and related methods IAPP, GIPR, INSR CYP3A4 4563/4885ALDH1A1 4542/4885MAPT 1706/4885
US-10596300-B2 Methods and compositions relating to biocompatible implants CD44, ILK, CRYAA CYP3A4 3428/4885ALDH1A1 1067/4885MAPT 4224/4885
US-20220125937-A1 ZWITTERIONIC POLYMER-INSULIN COMPOSITIONS AND RELATED METHODS IAPP, INSR, IRS1 CYP3A4 4617/4885ALDH1A1 4850/4885MAPT 1304/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.