SCHEMBL4616965

SCHEMBL4616965

COc1cccc(S(=O)(=O)F)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 6/20 0.53
KEAP1 Q14145 3/20 0.53
FFAR4 Q5NUL3 1/20 0.53
PGR P06401 4/20 0.53
TAS2R14 Q9NYV8 1/20 0.51
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
MEP1B Q16820 1/20 0.49
MET P08581 1/20 0.48
GAA P10253 1/20 0.48
ACHE P22303 1/20 0.47
LMNA P02545 1/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31352975 0.83 MTNR1B (0.56) NFE2L2KEAP1FFAR4PGRCA12
SCHEMBL3151230 0.83 MTNR1B (0.56) NFE2L2KEAP1FFAR4PGRCA12
SCHEMBL29650302 0.82 NFE2L2 (0.54) NFE2L2KEAP1FFAR4PGRTAS2R14
SCHEMBL803706 0.82 NFE2L2 (0.54) NFE2L2KEAP1FFAR4PGRTAS2R14
SCHEMBL11155550 0.82 NFE2L2 (0.54) NFE2L2KEAP1FFAR4PGRTAS2R14
SCHEMBL29782844 0.81 PGR (0.61) NFE2L2KEAP1FFAR4PGRTAS2R14
SCHEMBL4952964 0.81 PGR (0.61) NFE2L2KEAP1FFAR4PGRTAS2R14
SCHEMBL13290766 0.80 NFE2L2 (0.53) NFE2L2KEAP1FFAR4PGRTAS2R14
SCHEMBL18152 0.80 NFE2L2 (0.53) NFE2L2KEAP1FFAR4PGRTAS2R14
SCHEMBL2377950 0.80 NFE2L2 (0.53) NFE2L2KEAP1FFAR4PGRTAS2R14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119219808-A Multifunctional ionic polymer, preparation method and application thereof, and ion exchange membrane 佛山绿动氢能科技有限公司 2024-12-31 CN disclosed
US-20080318933-A1 5-Sulfonyl-1-Piperidinyl Substituted Indole Derivatives as 5-Ht6 Receptor Antagonists for the Treatment of Cns Disorders GLAXO GROUP LIMITED 2008-12-25 US disclosed
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP disclosed
EP-1814873-A2 5-SULFONYL-1-PIPERIDINYL SUBSTITUTED INDOLE DERIVATIVES AS 5-HT6 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF CNS DISORDERS GLAXO GROUP LIMITED (GB) 2007-08-08 EP disclosed
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof WYETH (US) 2006-12-07 US disclosed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO disclosed
WO-2006038006-A2 5-SULFONYL-1-PIPERIDINYL SUBSTITUTED INDOLE DERIVATIVES AS 5-HT6 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF CNS DISORDERS GLAXO GROUP LIMITED (GB) 2006-04-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080318933-A1 5-Sulfonyl-1-Piperidinyl Substituted Indole Derivatives as 5-Ht6 Receptor Antagonists for the Treatment of Cns Disorders HTR6, HTR5A, TPH1 NFE2L2 3671/4885KEAP1 2343/4885FFAR4 186/4885
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof SFRP1, SOS1, FZD7 NFE2L2 3293/4885KEAP1 1841/4885FFAR4 1926/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.