SCHEMBL4624470

SCHEMBL4624470

CC(C)OC(=O)C(C#N)=C([O-])C(F)(F)F.[Na+]

nearest known ligand 0.39

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.39
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4625275 0.81 IDO1 (0.36) ALDH1A1
SCHEMBL4624472 0.78 HPGD (0.40) HPGDALDH1A1
SCHEMBL4624468 0.78 HPGD (0.40) HPGDALDH1A1
SCHEMBL2592392 0.77 ALDH1A1 (0.44) ALDH1A1
SCHEMBL31735349 0.77 ALDH1A1 (0.44) ALDH1A1
SCHEMBL10991319 0.71 HPGD (0.44) HPGDALDH1A1
Potassium Ion SCHEMBL11036364 0.69 HPGD (0.43) HPGDALDH1A1
SCHEMBL11036370 0.69 HPGD (0.43) HPGDALDH1A1
Potassium Ion SCHEMBL11036367 0.67 HPGD (0.41) HPGDALDH1A1
SCHEMBL13007000 0.63 HPGD (0.42) HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1067121-B1 5-Aminopyrazole-4-carboxylate derivative and process for preparing the same MITSUI CHEMICALS INC (JP) 2008-05-28 EP disclosed
US-6235911-B1 5-aminopyrazole-4-carboxylate derivative and process for preparing the same MITSUI CHEMICALS, INC. (JP) 2001-05-22 US disclosed
EP-1067121-A2 5-Aminopyrazole-4-carboxylate derivative and process for preparing the same Mitsui Chemicals, Inc. (JP) 2001-01-10 EP disclosed