SCHEMBL4663552

SCHEMBL4663552

COc1ccccc1C1(O)CCC(c2ccccc2)CC1Cc1ccccc1N(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
SIGMAR1 Q99720 1/20 0.37
TACR1 P25103 8/20 0.35
GRIN2B Q13224 1/20 0.35
ATP1A1 P05023 2/20 0.35
ATP1B1 P05026 2/20 0.35
ATP1A3 P13637 2/20 0.35
ATP1B2 P14415 2/20 0.35
ATP1A2 P50993 2/20 0.35
ATP1B3 P54709 2/20 0.35
FXYD2 P54710 2/20 0.35
ATP1A4 Q13733 2/20 0.35
KDM1A O60341 3/20 0.34
MAOA P21397 3/20 0.34
MAOB P27338 2/20 0.34
NR3C1 P04150 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4665556 0.84 SIGMAR1 (0.39) CHRM2CHRM1SIGMAR1ATP1A1ATP1B1
SCHEMBL4667320 0.81 OPRK1 (0.50) CHRM2CHRM1OPRM1OPRD1OPRK1
SCHEMBL5719790 0.78 ATP1A1 (0.33) TACR1ATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL4664155 0.78 OPRK1 (0.38) CHRM2CHRM1TACR1ATP1A1ATP1B1
SCHEMBL4663722 0.75 MAOA (0.35) TACR1ATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL4664194 0.75 TACR1 (0.34) TACR1ATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL4667252 0.74 OPRM1 (0.37) SIGMAR1ATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL4663548 0.73 OPRM1 (0.41) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL4665510 0.72 SIGMAR1 (0.36) SIGMAR1ATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL6939500 0.71 SLC6A2 (0.47) CHRM2CHRM1SIGMAR1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1571140-B1 C-substituted cyclohexylmethylamine derivatives GRUENENTHAL GMBH (DE) 2008-11-12 EP claimed