SCHEMBL4663722

SCHEMBL4663722

CN(C)c1ccccc1CC1CC(c2ccccc2)CCC1(O)Cc1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.35
OPRL1 P41146 2/20 0.34
ATP1A1 P05023 3/20 0.33
ATP1B1 P05026 3/20 0.33
ATP1A3 P13637 3/20 0.33
ATP1B2 P14415 3/20 0.33
ATP1A2 P50993 3/20 0.33
ATP1B3 P54709 3/20 0.33
FXYD2 P54710 3/20 0.33
ATP1A4 Q13733 3/20 0.33
TRPA1 O75762 1/20 0.33
LMNA P02545 1/20 0.33
NPY2R P49146 2/20 0.31
KDM4E B2RXH2 1/20 0.31
EPHX2 P34913 1/20 0.31
OPRM1 P35372 1/20 0.30
OPRK1 P41145 1/20 0.30
AKR1C3 P42330 1/20 0.30
AKR1C1 Q04828 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4667252 0.89 OPRM1 (0.37) MAOAOPRL1ATP1A1ATP1B1ATP1A3
SCHEMBL4665510 0.87 SIGMAR1 (0.36) MAOAOPRL1ATP1A1ATP1B1ATP1A3
SCHEMBL6936768 0.81 SLC6A9 (0.39) MAOAOPRL1TRPA1LMNAOPRM1
Hydrochloric Acid SCHEMBL7741185 0.80 OPRL1 (0.39) MAOAOPRL1TRPA1LMNAOPRM1
SCHEMBL4664194 0.80 TACR1 (0.34) MAOAATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL4664155 0.75 OPRK1 (0.38) OPRL1ATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL4663552 0.75 CHRM2 (0.38) MAOAOPRL1ATP1A1ATP1B1ATP1A3
SCHEMBL5719790 0.75 ATP1A1 (0.33) MAOAATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL4665556 0.75 SIGMAR1 (0.39) OPRL1ATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL4667320 0.73 OPRK1 (0.50) OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1571140-B1 C-substituted cyclohexylmethylamine derivatives GRUENENTHAL GMBH (DE) 2008-11-12 EP claimed
EP-1043307-B1 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use GRUENENTHAL GMBH (DE) 2003-06-04 EP claimed
EP-1043307-A2 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use Grünenthal GmbH (DE) 2000-10-11 EP claimed
EP-1043307-B1 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use GRUENENTHAL GMBH (DE) 2003-06-04 EP disclosed
US-6410790-B1 ANALGESICS GRUENENTHAL GMBH (DE) 2002-06-25 US disclosed
EP-1043307-A2 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use Grünenthal GmbH (DE) 2000-10-11 EP disclosed