SCHEMBL4665556

SCHEMBL4665556

COc1ccc(C2(O)CCC(c3ccccc3)CC2Cc2ccccc2N(C)C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.39
OPRM1 P35372 5/20 0.38
OPRL1 P41146 3/20 0.38
SLC6A9 P48067 2/20 0.37
SLC6A4 P31645 4/20 0.36
SLC6A2 P23975 3/20 0.36
SLC22A1 O15245 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
OPRD1 P41143 2/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
OPRK1 P41145 1/20 0.36
CNR2 P34972 1/20 0.36
ATP1A1 P05023 1/20 0.35
ATP1B1 P05026 1/20 0.35
ATP1A3 P13637 1/20 0.35
ATP1B2 P14415 1/20 0.35
ATP1A2 P50993 1/20 0.35
ATP1B3 P54709 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4667320 0.89 OPRK1 (0.50) OPRM1SLC6A4SLC6A2SLC22A1MEN1
SCHEMBL5719790 0.86 ATP1A1 (0.33) OPRM1OPRD1CNR2ATP1A1ATP1B1
SCHEMBL4663552 0.84 CHRM2 (0.38) SIGMAR1OPRM1OPRL1OPRD1CHRM2
SCHEMBL6934477 0.82 SLC6A4 (0.52) OPRM1OPRL1SLC6A9SLC6A4SLC6A2
SCHEMBL4664155 0.82 OPRK1 (0.38) OPRM1OPRL1SLC6A4SLC6A2SLC22A1
SCHEMBL4663722 0.75 MAOA (0.35) OPRM1OPRL1OPRK1ATP1A1ATP1B1
SCHEMBL4664194 0.75 TACR1 (0.34) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2
SCHEMBL4667252 0.74 OPRM1 (0.37) SIGMAR1OPRM1OPRL1MEN1KMT2A
SCHEMBL4664132 0.73 OPRM1 (0.41) SIGMAR1OPRM1OPRL1SLC6A9SLC6A4
SCHEMBL4665510 0.72 SIGMAR1 (0.36) SIGMAR1OPRM1OPRL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1571140-B1 C-substituted cyclohexylmethylamine derivatives GRUENENTHAL GMBH (DE) 2008-11-12 EP claimed