SCHEMBL4667252

SCHEMBL4667252

CN(C)c1ccccc1CC1CC(c2ccccc2)CCC1(O)CCc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 5/20 0.37
OPRL1 P41146 4/20 0.37
MAOA P21397 2/20 0.34
OPRD1 P41143 2/20 0.34
OPRK1 P41145 2/20 0.34
SIGMAR1 Q99720 2/20 0.33
MEN1 O00255 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
ATP1A1 P05023 1/20 0.32
ATP1B1 P05026 1/20 0.32
ATP1A3 P13637 1/20 0.32
ATP1B2 P14415 1/20 0.32
ATP1A2 P50993 1/20 0.32
ATP1B3 P54709 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4665510 0.94 SIGMAR1 (0.36) OPRM1OPRL1MAOASIGMAR1MEN1
SCHEMBL4663722 0.89 MAOA (0.35) OPRM1OPRL1MAOAOPRK1CYP3A4
SCHEMBL6678803 0.82 OPRM1 (0.40) OPRM1OPRL1OPRD1OPRK1SLC18A3
SCHEMBL4664194 0.78 TACR1 (0.34) MAOACYP3A4CYP2D6ATP1A1ATP1B1
SCHEMBL6676478 0.76 SLC18A3 (0.40) OPRM1OPRL1OPRD1OPRK1SLC18A3
Hydrochloric Acid SCHEMBL7737765 0.75 SLC18A3 (0.39) OPRM1OPRL1OPRD1OPRK1SLC18A3
SCHEMBL4664155 0.74 OPRK1 (0.38) OPRM1OPRL1OPRD1OPRK1MEN1
SCHEMBL4663552 0.74 CHRM2 (0.38) OPRM1OPRL1MAOAOPRD1OPRK1
SCHEMBL5719790 0.74 ATP1A1 (0.33) OPRM1MAOAOPRD1ATP1A1ATP1B1
SCHEMBL4665556 0.74 SIGMAR1 (0.39) OPRM1OPRL1OPRD1OPRK1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1571140-B1 C-substituted cyclohexylmethylamine derivatives GRUENENTHAL GMBH (DE) 2008-11-12 EP claimed