SCHEMBL4694380

SCHEMBL4694380

NC(=O)c1ccccc1[CH]CCN1CC2CN(Cc3ccc(Cl)c(Cl)c3)C[C@@H]2C1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.41
SIGMAR1 Q99720 5/20 0.41
CCR2 P41597 1/20 0.40
S1PR5 Q9H228 4/20 0.40
S1PR1 P21453 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
HTR2A P28223 1/20 0.39
KCNH2 Q12809 1/20 0.39
CCR3 P51677 2/20 0.38
CACNA1G O43497 1/20 0.38
HTT P42858 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3282844 0.88 GRIN2B (0.44) S1PR5S1PR1DRD2KCNH2
SCHEMBL4694985 0.88 GRIN2B (0.44) S1PR5S1PR1DRD2KCNH2
SCHEMBL4689903 0.80 P2RX7 (0.41) MEN1KMT2AHTTALDH1A1
SCHEMBL4691802 0.78 CCR5 (0.48) MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL3284078 0.77 CHRNA4 (0.39) KDM4E
SCHEMBL4692840 0.76 PARP1 (0.40) KMT2ADRD2KDM4EALDH1A1
SCHEMBL4694455 0.75 CHRNB2 (0.44) MEN1KMT2AKCNH2ALDH1A1SMN1; SMN2
SCHEMBL4693059 0.75 CCR5 (0.37) MEN1KMT2AKDM4EALDH1A1
SCHEMBL4694264 0.75 ALDH1A1 (0.36) ALDH1A1
SCHEMBL3284141 0.75 CCR5 (0.42) SIGMAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed