SCHEMBL4690544

SCHEMBL4690544

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4ccc(N(C)CCO)cc4)CC3C2)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.35
HPGD P15428 1/20 0.34
CCR5 P51681 3/20 0.34
KDM1A O60341 1/20 0.33
TNF P01375 1/20 0.33
UBE2M P61081 1/20 0.33
DCUN1D1 Q96GG9 1/20 0.33
SLC6A2 P23975 4/20 0.32
SLC6A4 P31645 4/20 0.32
SLC6A3 Q01959 3/20 0.32
ALDH1A1 P00352 2/20 0.32
POLB P06746 1/20 0.32
PARP1 P09874 1/20 0.32
PARP2 Q9UGN5 1/20 0.32
S1PR1 P21453 1/20 0.32
CNR2 P34972 2/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
OPRK1 P41145 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692070 0.90 HPGD (0.36) HPGDCCR5KDM1ATNFUBE2M
SCHEMBL4695972 0.84 CHRNB2 (0.40) HPGDTNFALDH1A1POLBHCRTR1
SCHEMBL4689519 0.83 ALDH1A1 (0.47) HPGDTNFALDH1A1POLBHCRTR1
SCHEMBL4695951 0.83 LMNA (0.39) HPGDTNFPOLBHCRTR1HCRTR2
SCHEMBL4693590 0.82 KDM1A (0.48) KDM1AALDH1A1
SCHEMBL4690534 0.82 LMNA (0.39) L3MBTL1HPGDTNFCNR2
SCHEMBL4690843 0.82 GAA (0.41) HPGDSLC6A4
SCHEMBL4691641 0.80 CHRNB2 (0.43) L3MBTL1HPGDCCR5TNFALDH1A1
SCHEMBL4694328 0.80 TNF (0.35) HPGDKDM1ATNFALDH1A1POLB
SCHEMBL4690738 0.79 HCRTR1 (0.46) HPGDTNFALDH1A1HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed