SCHEMBL4698653

SCHEMBL4698653

CCCC[C@H](NC(=O)N[C@@H](CC(=O)O)c1ccc2c(c1)OCO2)C(=O)N1CCN(C(=O)c2cccs2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.47
ALDH1A1 P00352 3/20 0.42
GAA P10253 2/20 0.42
ITGB3 P05106 6/20 0.41
ITGA2B P08514 5/20 0.41
ITGAV P06756 3/20 0.41
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HPGD P15428 2/20 0.40
POLB P06746 1/20 0.40
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
F2R P25116 1/20 0.39
TAS1R3 Q7RTX0 2/20 0.38
TAS1R1 Q7RTX1 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
F2 P00734 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4702813 0.89 ALDH1A1 (0.45) LMNAALDH1A1GAAITGB3ITGA2B
SCHEMBL4701238 0.87 PKM (0.45) ALDH1A1GAAITGB3ITGA2BHPGD
SCHEMBL7900498 0.83 CCR1 (0.46) GAAITGB3ITGA2BITGAVF2R
SCHEMBL4701810 0.82 ALDH1A1 (0.44) ALDH1A1GAAITGB3ITGA2BITGAV
SCHEMBL4701020 0.82 P2RY12 (0.43) GAAITGB3ITGA2BITGAVTAS1R3
SCHEMBL4698338 0.81 ALDH1A1 (0.47) LMNAALDH1A1GAACYP2D6CYP2C9
SCHEMBL7892913 0.81 ITGB3 (0.40) LMNAALDH1A1GAAITGB3ITGA2B
SCHEMBL7955769 0.80 HPGD (0.47) GAAITGB3ITGA2BITGAVHPGD
SCHEMBL7904100 0.80 ITGB3 (0.41) LMNAGAAITGB3ITGA2BITGAV
SCHEMBL20530282 0.80 POLB (0.46) GAAITGB3ITGA2BITGAVHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1071680-B1 N,N-DISUBSTITUTED AMIDES THAT INHIBIT THE BINDING OF INTEGRINS TO THEIR RECEPTORS ENCYSIVE PHARMACEUTICALS INC (US) 2008-07-23 EP disclosed
US-6194448-B1 ANTIINFLAMMATORY AGENTS; ASTHMA; RHEUMATIC DISORDERS TEXAS BIOTECHNOLOGY CORPORATION 2001-02-27 US disclosed