SCHEMBL4701810

SCHEMBL4701810

CCCC[C@H](NC(=O)N[C@@H](CC(=O)O)c1ccc2c(c1)OCO2)C(=O)N1CCN(Cc2ccsc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.44
KDM4E B2RXH2 7/20 0.44
TDP1 Q9NUW8 3/20 0.41
POLB P06746 2/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
ITGB3 P05106 4/20 0.40
ITGA2B P08514 3/20 0.40
HTT P42858 1/20 0.40
ITGAV P06756 1/20 0.39
GAA P10253 2/20 0.39
MCHR1 Q99705 2/20 0.38
MAPT P10636 1/20 0.38
F2R P25116 1/20 0.38
FAAH O00519 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4702813 0.87 ALDH1A1 (0.45) ALDH1A1KDM4EPOLBKMT2AMEN1
SCHEMBL7900328 0.84 ALDH1A1 (0.43) ALDH1A1KDM4ETDP1POLBKMT2A
SCHEMBL7900090 0.83 GAA (0.41) KMT2AITGB3ITGA2BITGAVGAA
SCHEMBL4698653 0.82 LMNA (0.47) ALDH1A1POLBITGB3ITGA2BITGAV
SCHEMBL7900104 0.81 APOBEC3A (0.47) ALDH1A1KDM4ETDP1KMT2AMEN1
SCHEMBL4701020 0.81 P2RY12 (0.43) ITGB3ITGA2BITGAVGAA
SCHEMBL4701238 0.80 PKM (0.45) ALDH1A1POLBKMT2AMEN1ITGB3
SCHEMBL7900498 0.79 CCR1 (0.46) ITGB3ITGA2BITGAVGAAF2R
SCHEMBL4698338 0.79 ALDH1A1 (0.47) ALDH1A1KDM4EKMT2AMEN1GAA
SCHEMBL7892913 0.78 ITGB3 (0.40) ALDH1A1ITGB3ITGA2BITGAVGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1071680-B1 N,N-DISUBSTITUTED AMIDES THAT INHIBIT THE BINDING OF INTEGRINS TO THEIR RECEPTORS ENCYSIVE PHARMACEUTICALS INC (US) 2008-07-23 EP disclosed
US-6194448-B1 ANTIINFLAMMATORY AGENTS; ASTHMA; RHEUMATIC DISORDERS TEXAS BIOTECHNOLOGY CORPORATION 2001-02-27 US disclosed