Furan-3-Carbaldehyde

Furan-3-Carbaldehyde

SCHEMBL4740464

O=Cc1ccoc1.O=S([O-])O.[Na+]

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Furan-3-Carbaldehyde. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 known ✓ P09917 2/20 0.35
HCAR2 Q8TDS4 1/20 0.43
ERN1 O75460 5/20 0.35
MAPT P10636 2/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 4/20 0.34
TDP1 Q9NUW8 2/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
DNMT1 P26358 1/20 0.33
DUSP3 P51452 1/20 0.33
PTPN5 P54829 1/20 0.33
PTPN11 Q06124 1/20 0.33
MCL1 Q07820 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP1B1 Q16678 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Furan-3-Carbaldehyde SCHEMBL133204 0.83
Furan-3-Carbaldehyde SCHEMBL27487877 0.81
Furan-3-Carbaldehyde SCHEMBL27570297 0.77 HCAR2 (0.45) HCAR2ERN1MAPTALOX5ALDH1A1
Furan-3-Carbaldehyde SCHEMBL12006489 0.74 HCAR2 (0.42) HCAR2ERN1MAPTALOX5ALDH1A1
Furan-3-Carbaldehyde SCHEMBL8212634 0.72 HCAR2 (0.50) HCAR2ERN1MAPTALOX5ALDH1A1
Benzaldehyde SCHEMBL9452552 0.71 ALDH1A1 (0.64) HCAR2MAPTALOX5ALDH1A1KMT2A
Benzaldehyde SCHEMBL29105107 0.71 ALDH1A1 (0.64) HCAR2MAPTALOX5ALDH1A1KMT2A
Furan-3-Carbaldehyde SCHEMBL12006488 0.69 HCAR2 (0.39) HCAR2ERN1MAPTALOX5ALDH1A1
Sulfurous Acid SCHEMBL28112791 0.68 ALDH5A1 (0.43) ERN1ALDH1A1
Benzaldehyde SCHEMBL9258080 0.68 ALDH1A1 (0.58) HCAR2MAPTALOX5ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008081266-A1 COMPOUNDS FOR THE TREATMENT OR PREVENTION OF INFECTION BY FLAVIVIRIDAE CARTA ANTONIO (IT) 2008-07-10 WO disclosed