SCHEMBL4752455

SCHEMBL4752455

CCC(Oc1cc(Cl)cc2c1OC(C)(C)C2)N1CCC(n2c(=O)[nH]c3ccc(Cl)cc32)CC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 19/20 0.47
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
SLC6A4 P31645 1/20 0.43
DRD3 P35462 1/20 0.43
OPRL1 P41146 4/20 0.39
CACNA1F O60840 1/20 0.38
CHRM1 P11229 1/20 0.38
ADRA1D P25100 1/20 0.38
HTR7 P34969 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
CACNA1D Q01668 1/20 0.38
CACNA1S Q13698 1/20 0.38
CACNA1C Q13936 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4750828 0.94 HTR1A (0.51) OPRM1HTR1AADRA2ADRD2HTR2A
Hydrochloric Acid SCHEMBL4817572 0.88 OPRM1 (0.45) OPRM1HTR1AADRA2ADRD2HTR2A
SCHEMBL4754005 0.81 DRD2 (0.42) OPRM1DRD2SLC6A4OPRL1OPRD1
SCHEMBL4754022 0.81 OPRM1 (0.49) OPRM1HTR1AADRA2ADRD2HTR2A
SCHEMBL4752471 0.79 OPRM1 (0.42) OPRM1HTR1ADRD2HTR2ADRD3
SCHEMBL4750799 0.77 POLB (0.42) HTR2A
SCHEMBL4753001 0.76 DRD2 (0.58) OPRM1HTR1AADRA2ADRD2HTR2A
SCHEMBL4750861 0.76 PLD2 (0.45) OPRM1DRD2OPRL1
Water SCHEMBL4912684 0.74 OPRL1 (0.52) OPRM1DRD2OPRL1CHRM1
SCHEMBL4855972 0.73 OPRL1 (0.65) OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008146064-A1 NEW BENZOFURAN DERIVATIVES AS SELECTIVE 5HT7 RECEPTOR INHIBITORS AND PROCESS FOR THEIR PREPARATION EGIS GYÓGYSZERGYÁR (HU) 2008-12-04 WO disclosed