Ethanesulfonic Acid Amide

Ethanesulfonic Acid Amide

SCHEMBL4800715

CCS(N)(=O)=O.Cc1cc(C)cc(C)c1

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
KDM4E B2RXH2 1/20 0.48
TSHR P16473 2/20 0.45
CA2 P00918 9/20 0.40
CA1 P00915 8/20 0.40
CA9 Q16790 7/20 0.40
CA12 O43570 3/20 0.40
CA6 P23280 2/20 0.40
CA5A P35218 2/20 0.40
CA7 P43166 2/20 0.40
CA5B Q9Y2D0 2/20 0.40
CA3 P07451 1/20 0.40
CYP3A4 P08684 1/20 0.39
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
RAPGEF4 Q8WZA2 1/20 0.37
CA4 P22748 1/20 0.36
CA13 Q8N1Q1 1/20 0.36
CA14 Q9ULX7 1/20 0.36
TPMT P51580 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfamide SCHEMBL29026073 0.84 ALDH1A1 (0.55) ALDH1A1KDM4ETSHRCA2CA1
Methanesulfonamide SCHEMBL4804491 0.81 CA1 (0.53) ALDH1A1KDM4ETSHRCA2CA1
Methanesulfonamide SCHEMBL4804172 0.81 CA1 (0.53) ALDH1A1KDM4ETSHRCA2CA1
SCHEMBL4878731 0.79 CA1 (0.48) ALDH1A1KDM4ETSHRCA2CA1
Ethanesulfonic Acid Amide SCHEMBL28038 0.77
Toluene SCHEMBL303284 0.76 ACHE (0.55) TSHRCA2CA1CA9CA12
SCHEMBL2005577 0.74 CA2 (0.56) ALDH1A1KDM4ETSHRCA2CA1
Ethylamine SCHEMBL29162867 0.74 ALDH1A1 (0.56) ALDH1A1TSHRTPMTPRSS1PRSS2
Ethanesulfonic Acid Amide SCHEMBL27415310 0.74 CA2 (0.46) CA2CA1CA9CA12CA6
Ethanesulfonic Acid Amide SCHEMBL3402460 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7414154-B2 Polyamine compounds and compositions for use in conjunction with cancer therapy WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2008-08-19 US disclosed
US-7314959-B2 Amino thiol compounds and compositions for use in conjunction with cancer therapy WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2008-01-01 US disclosed
US-20050101676-A1 Amino thiol compounds and compositions for use in conjunction with cancer therapy NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2005-05-12 US disclosed
WO-2005014524-A2 AMINO THIOL COMPOUNDS AND COMPOSITIONS FOR USE IN CONJUNCTION WITH CANCER THERAPY WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2005-02-17 WO disclosed
US-20050027016-A1 Polyamine compounds and compositions for use in conjection with cancer therapy FAHL KATHLEEN L (US) 2005-02-03 US disclosed
EP-1478618-A1 POLYAMINE COMPOUNDS AND COMPOSITIONS FOR USE IN CONJUNCTION WITH CANCER THERAPY WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2004-11-24 EP disclosed
US-20040225021-A1 Polyamine compounds and compositions for use in conjunction with cancer therapy WISCONSIN ALUMNI RESEARCH FOUNDATION 2004-11-11 US disclosed
US-20030185778-A1 Polyamine compounds and compositions for use in conjunction with cancer therapy NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-10-02 US disclosed
WO-2003066572-A1 POLYAMINE COMPOUNDS AND COMPOSITIONS FOR USE IN CONJUNCTION WITH CANCER THERAPY WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2003-08-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040225021-A1 Polyamine compounds and compositions for use in conjunction with cancer therapy SRM, SMS, HNMT ALDH1A1 926/4885KDM4E 1966/4885TSHR 4317/4885
US-20050101676-A1 Amino thiol compounds and compositions for use in conjunction with cancer therapy SRM, MGMT, AADAT ALDH1A1 692/4885KDM4E 2612/4885TSHR 3537/4885
US-20050027016-A1 Polyamine compounds and compositions for use in conjection with cancer therapy SRM, SMS, SMOX ALDH1A1 1265/4885KDM4E 2972/4885TSHR 4150/4885
US-20030185778-A1 Polyamine compounds and compositions for use in conjunction with cancer therapy SRM, SMS, HNMT ALDH1A1 926/4885KDM4E 1966/4885TSHR 4317/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.