Dicloxacillin

Dicloxacillin

SCHEMBL4928524

Cc1onc(-c2c(Cl)cccc2Cl)c1C(=O)N[C@@H]1C(=O)N2[C@@H]1SC(C)(C)[C@@H]2C(=O)O.O

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

mecApbp2pbp4pbpApbpF

The experimentally established mechanism targets of Dicloxacillin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 4/20 0.98
CYP1A2 P05177 1/20 0.89
SLCO1B3 Q9NPD5 1/20 0.84
SLCO1B1 Q9Y6L6 1/20 0.84
LMNA P02545 4/20 0.82
HPGD P15428 3/20 0.82
TDP1 Q9NUW8 2/20 0.82
MEN1 O00255 1/20 0.82
KMT2A Q03164 1/20 0.82
ALDH1A1 P00352 1/20 0.66
SMN1; SMN2 Q16637 1/20 0.66
PTGS1 P23219 1/20 0.58
PDE3A Q14432 1/20 0.58
KDM4E B2RXH2 1/20 0.49
TSHR P16473 1/20 0.49
RECQL P46063 1/20 0.49
HRH1 P35367 1/20 0.49
SLC22A8 Q8TCC7 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dicloxacillin SCHEMBL5595924 1.00 ABCB11 (0.98) ABCB11CYP1A2SLCO1B3SLCO1B1LMNA
Dicloxacillin SCHEMBL5549845 0.99 ABCB11 (0.97) ABCB11CYP1A2SLCO1B3SLCO1B1LMNA
Dicloxacillin SCHEMBL11407716 0.99 ABCB11 (1.00) ABCB11CYP1A2SLCO1B3SLCO1B1LMNA
Dicloxacillin SCHEMBL11407710 0.99 ABCB11 (1.00) ABCB11CYP1A2SLCO1B3SLCO1B1LMNA
Dicloxacillin SCHEMBL11407708 0.99 ABCB11 (1.00) ABCB11CYP1A2SLCO1B3SLCO1B1LMNA
Dicloxacillin SCHEMBL8727180 0.99 ABCB11 (1.00) ABCB11CYP1A2SLCO1B3SLCO1B1LMNA
Dicloxacillin SCHEMBL23955 0.99 ABCB11 (1.00) ABCB11CYP1A2SLCO1B3SLCO1B1LMNA
Dicloxacillin SCHEMBL41517 0.98 ABCB11 (0.98) ABCB11CYP1A2SLCO1B3SLCO1B1LMNA
Dicloxacillin SCHEMBL28540896 0.98 ABCB11 (0.98) ABCB11CYP1A2SLCO1B3SLCO1B1LMNA
Dicloxacillin SCHEMBL28536434 0.98 ABCB11 (0.98) ABCB11CYP1A2SLCO1B3SLCO1B1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080139545-A1 FORMULATION TO TREAT EAR INFECTION CHOE WON-TAEK 2008-06-12 US disclosed
EP-1827408-A1 METHOD FOR TREATING SKIN DISORDERS WITH XANTHOPHYLLS Nu-Tein Co., Inc. (US) 2007-09-05 EP disclosed
EP-1827400-A2 TOPICAL SKIN PATCH CONTAINING XANTHOPHYLLS Nu-Tein Co., Inc. (US) 2007-09-05 EP disclosed
EP-1814540-A2 COMPOSITIONS USEFUL TO TREAT OCULAR NEOVASCULAR DISEASES AND MACULAR DEGENERATION Nu-Tein Co., Inc. (US) 2007-08-08 EP disclosed
US-20060134226-A1 Compositions useful to treat ocular neovascular diseases and macular degeneration NU-TEIN CO., LTD. 2006-06-22 US disclosed
WO-2006062740-A2 TOPICAL SKIN PATCH CONTAINING XANTHOPHYLLS NU-TEIN CO., INC. (US) 2006-06-15 WO disclosed
WO-2006060475-A1 METHOD FOR TREATING SKIN DISORDERS WITH XANTHOPHYLLS NU-TEIN CO., INC. (US) 2006-06-08 WO disclosed
US-20060122282-A1 METHOD FOR TREATING SKIN DISORDERS WITH XANTHOPHYLLS NU-TEIN CO., INC. 2006-06-08 US disclosed
WO-2006055526-A2 COMPOSITIONS USEFUL TO TREAT OCULAR NEOVASCULAR DISEASES AND MACULAR DEGENERATION NU-TEIN CO., INC. (US) 2006-05-26 WO disclosed
US-20050089473-A1 Potassium channel mediated delivery of agents through the blood-brain barrier CEDARS-SINAI MEDICAL CENTER 2005-04-28 US disclosed
US-20020042394-A1 Cobalamin compounds useful as antibiotic agents and as imaging agents HOGENKAMP HENRICUS P C (US) 2002-04-11 US disclosed
WO-2001092288-A2 COBALAMIN COMPOUNDS USEFUL AS ANTIBIOTIC AGENTS AND AS IMAGING AGENTS MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2001-12-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060134226-A1 Compositions useful to treat ocular neovascular diseases and macular degeneration CFD, VEGFA, CFH ABCB11 3768/4885CYP1A2 2767/4885SLCO1B3 1727/4885
US-20050089473-A1 Potassium channel mediated delivery of agents through the blood-brain barrier KCNN2, KCNN1, KCNN3 ABCB11 218/4885CYP1A2 4314/4885SLCO1B3 290/4885
US-20020042394-A1 Cobalamin compounds useful as antibiotic agents and as imaging agents MMAB, BLVRB, AHCY ABCB11 100/4885CYP1A2 1391/4885SLCO1B3 104/4885
US-20060122282-A1 METHOD FOR TREATING SKIN DISORDERS WITH XANTHOPHYLLS COL1A1, COL2A1, KRT18 ABCB11 558/4885CYP1A2 1109/4885SLCO1B3 3566/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.