SCHEMBL493466

SCHEMBL493466

CN(C)c1ccccc1CC1CCC(CNC(=O)COC2CCCN(S(=O)(=O)c3c(Cl)cc(Cl)cc3Cl)C2)CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
MAPT P10636 3/20 0.37
USP2 O75604 1/20 0.37
TP53 P04637 3/20 0.37
THRB P10828 1/20 0.37
FAAH O00519 1/20 0.35
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
JAK3 P52333 1/20 0.35
EPHX2 P34913 1/20 0.34
ACLY P53396 1/20 0.34
ATM Q13315 1/20 0.34
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL493066 0.91 RAB9A (0.39) LMNAMAPTUSP2TP53THRB
SCHEMBL3661024 0.86 TRPV4 (0.39) TP53FAAHBCHEACHEEPHX2
SCHEMBL493760 0.86 PKM (0.37) LMNAEPHX2ACLYATM
SCHEMBL493465 0.84 KMT2A (0.37) LMNAMAPTUSP2TP53THRB
SCHEMBL493203 0.80 FAAH (0.37) LMNATP53THRBFAAHBCHE
SCHEMBL493302 0.79 FAAH (0.39) LMNAFAAHBCHEACHEACLY
SCHEMBL493619 0.78 KMT2A (0.37) LMNAUSP2THRBFAAHBCHE
SCHEMBL493407 0.77 FAAH (0.37) LMNAFAAHBCHEACHEACLY
SCHEMBL3660998 0.77 ALDH1A1 (0.40) LMNAMAPTEPHX2
SCHEMBL492870 0.76 FAAH (0.38) FAAHBCHEACHEEPHX2ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106055-B2 Substituted amide compounds GRUENENTHAL GMBH (DE) 2012-01-31 US claimed
US-20080306084-A1 Substituted Amide Compounds GRUENENTHAL GMBH (DE) 2008-12-11 US claimed
US-8106055-B2 Substituted amide compounds GRUENENTHAL GMBH (DE) 2012-01-31 US disclosed
US-20080306084-A1 Substituted Amide Compounds GRUENENTHAL GMBH (DE) 2008-12-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080306084-A1 Substituted Amide Compounds OPRK1, NAA50, ACMSD LMNA 2485/4885MAPT 1653/4885USP2 4237/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.