SCHEMBL493680

SCHEMBL493680

O=C(O)COc1ccccc1NCS(=O)(=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
PTGDR2 Q9Y5Y4 11/20 0.47
ACLY P53396 3/20 0.45
CCR2 P41597 3/20 0.44
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CCR4 P51679 2/20 0.41
CCR5 P51681 2/20 0.41
KCNH2 Q12809 1/20 0.41
PTPN1 P18031 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Clamidoxic Acid SCHEMBL525147 0.73 KDM4E (0.54) ALDH1A1KCNH2
SCHEMBL493681 0.72 KMT2A (0.50) ALDH1A1PTGDR2PTPN1
SCHEMBL5516797 0.72 L3MBTL1 (0.56) ALDH1A1PTGDR2CYP2C19
SCHEMBL3531555 0.70 HTR1A (0.39) ALDH1A1CYP1A2CYP2C19
SCHEMBL1333288 0.69 PTGDR2 (0.56) PTGDR2ACLY
SCHEMBL1333486 0.68 PTGDR2 (0.67) ALDH1A1PTGDR2
SCHEMBL1331609 0.68 PTGDR2 (0.62) PTGDR2CYP2C19
SCHEMBL11223161 0.68 ALDH1A1 (0.57) ALDH1A1PTGDR2
SCHEMBL6165389 0.67 TDP1 (0.64) PTGDR2CYP2C19PTPN1
SCHEMBL101520 0.67 PTGDR2 (0.68) ALDH1A1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8580965-B2 Substituted sulfonamide compounds GRUENENTHAL GMBH (DE) 2013-11-12 US disclosed
US-8106055-B2 Substituted amide compounds GRUENENTHAL GMBH (DE) 2012-01-31 US disclosed
US-20080306084-A1 Substituted Amide Compounds GRUENENTHAL GMBH (DE) 2008-12-11 US disclosed
US-20080249128-A1 Substituted Sulfonamide Compounds GRUENENTHAL GMBH (DE) 2008-10-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080249128-A1 Substituted Sulfonamide Compounds BDKRB1, BDKRB2, NPSR1 ALDH1A1 2737/4885PTGDR2 74/4885ACLY 4105/4885
US-20080306084-A1 Substituted Amide Compounds OPRK1, NAA50, ACMSD ALDH1A1 1349/4885PTGDR2 135/4885ACLY 80/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.