Known targets — ChEMBL curated mechanism
ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO
The experimentally established mechanism targets of Sulfotep. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.
Predicted protein targets (top 16)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | CA1 known ✓ | P00915 | 1/20 | 0.30 |
| ▸ | TSHR | P16473 | 2/20 | 0.33 |
| ▸ | ALDH1A1 | P00352 | 1/20 | 0.33 |
| ▸ | CYP3A4 | P08684 | 1/20 | 0.33 |
| ▸ | MAPK1 | P28482 | 1/20 | 0.33 |
| ▸ | HSD17B10 | Q99714 | 1/20 | 0.33 |
| ▸ | MEN1 | O00255 | 1/20 | 0.32 |
| ▸ | KMT2A | Q03164 | 1/20 | 0.32 |
| ▸ | TDP1 | Q9NUW8 | 1/20 | 0.32 |
| ▸ | ALOX15 | P16050 | 1/20 | 0.32 |
| ▸ | FFAR3 | O14843 | 1/20 | 0.32 |
| ▸ | HDAC3 | O15379 | 1/20 | 0.32 |
| ▸ | HDAC1 | Q13547 | 1/20 | 0.32 |
| ▸ | HDAC2 | Q92769 | 1/20 | 0.32 |
| ▸ | HDAC8 | Q9BY41 | 1/20 | 0.32 |
| ▸ | PPARD | Q03181 | 1/20 | 0.31 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| Sulfotep SCHEMBL8781592 | 0.96 | ALOX15 (0.34) | TSHRALDH1A1CYP3A4MAPK1HSD17B10 | |
| Sulfotep SCHEMBL21925702 | 0.92 | ALOX15 (0.34) | TSHRALDH1A1CYP3A4MAPK1HSD17B10 | |
| Sulfotep SCHEMBL1419342 | 0.88 | ALOX15 (0.34) | TSHRALDH1A1CYP3A4MAPK1HSD17B10 | |
| Sulfotep SCHEMBL11362244 | 0.88 | MEN1 (0.34) | TSHRALDH1A1CYP3A4MAPK1HSD17B10 | |
| Sulfotep SCHEMBL4498444 | 0.86 | MEN1 (0.33) | TSHRALDH1A1CYP3A4MAPK1HSD17B10 | |
| Sulfotep SCHEMBL3695477 | 0.86 | MEN1 (0.33) | TSHRALDH1A1CYP3A4MAPK1HSD17B10 | |
| Sulfotep SCHEMBL19810563 | 0.85 | ALDH1A1 (0.34) | TSHRALDH1A1CYP3A4MAPK1HSD17B10 | |
| Sulfotep SCHEMBL8471621 | 0.84 | ALOX15 (0.37) | TSHRALDH1A1CYP3A4MAPK1HSD17B10 | |
| Sulfotep SCHEMBL53003 | 0.84 | ALOX15 (0.37) | TSHRALDH1A1CYP3A4MAPK1HSD17B10 | |
| Sulfotep SCHEMBL11870183 | 0.82 | ALOX15 (0.36) | TSHRALDH1A1CYP3A4MAPK1HSD17B10 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-3019554-B1 | A BINARY PROCESS FOR MANUFACTURE OF DIPPED LATEX PRODUCTS | TTK HEALTHCARE LTD (IN) | 2020-11-25 | — | — | EP | claimed |
| US-20160145401-A1 | BINARY PROCESS FOR MANUFACTURE OF DIPPED LATEX PRODUCTS | TKK Protective Devices Limited (IN) | 2016-05-26 | — | — | US | claimed |
| EP-3019554-A1 | A BINARY PROCESS FOR MANUFACTURE OF DIPPED LATEX PRODUCTS | Ttk Protective Devices Limited (IN) | 2016-05-18 | — | — | EP | claimed |
| EP-1986553-B1 | U-SHAPED DISC-SHUNT AND DELIVERY DEVICE | ALEEVA MEDICAL INC (US) | 2016-03-30 | — | — | EP | claimed |
| WO-2015004674-A1 | A BINARY PROCESS FOR MANUFACTURE OF DIPPED LATEX PRODUCTS | TTK PROTECTIVE DEVICES LIMITED (IN) | 2015-01-15 | — | — | WO | claimed |
| US-8361007-B2 | U-shaped disc shunt and delivery device | ALEEVA MEDICAL INC. (US) | 2013-01-29 | — | — | US | claimed |
| US-20090024071-A1 | U-Shaped Disc Shunt and Delivery Device | YEUNG JEFFREY E | 2009-01-22 | — | — | US | claimed |
| EP-1986553-A2 | U-SHAPED DISC-SHUNT AND DELIVERY DEVICE | Aleeva Medical, Inc. (US) | 2008-11-05 | — | — | EP | claimed |
| WO-2007089947-A2 | U-SHAPED DISC-SHUNT AND DELIVERY DEVICE | ALEEVA MEDICAL INC. (US) | 2007-08-09 | — | — | WO | claimed |
| US-20070169911-A1 | U-shaped disc shunt and delivery device | ALEEVA MEDICAL INC., A DELAWARE CORPORATION | 2007-07-26 | — | — | US | claimed |
| US-20070142791-A1 | U-shaped disc shunt and delivery device | ALEEVE MEDICAL INC. A DELAWARE CORPORATION | 2007-06-21 | — | — | US | claimed |
| CN-115944881-B | Heavy metal chelating agent for waste incineration fly ash and application method thereof | 合肥市东方美捷分子材料技术有限公司 | 2024-06-04 | — | — | CN | disclosed |
| EP-3497060-B1 | SYNTHETIC HYDROTALCITE | HEUBACH COLOUR PVT LTD (IN) | 2020-07-29 | — | — | EP | disclosed |
| EP-3497060-A2 | A SYNTHETIC HYDROTALCITE AND ONE PACK STABILIZER SYSTEM COMPRISING THE SAME | Heubach Colour Pvt. Ltd. (IN) | 2019-06-19 | — | — | EP | disclosed |
| WO-2018029704-A2 | A SYNTHETIC HYDROTALCITE AND ONE PACK STABILIZER SYSTEM COMPRISING THE SAME | HEUBACH COLOUR PVT. LTD. (IN) | 2018-02-15 | — | — | WO | disclosed |
| US-20060115738-A1 | Lithium-fluorinated carbon cells | WELLS FARGO BANK, NATIONAL ASSOCIATION | 2006-06-01 | — | — | US | disclosed |
| US-5298569-A | Time release agent polymers with main and side chains | NIPPON PAINT CO. (JP) | 1994-03-29 | — | — | US | disclosed |
| EP-0497758-A1 | FUNCTIONALIZED COPOLYMERS OF PARA-ALKYLSTYRENE/ISOOLEFIN PREPARED BY NUCLEOPHILIC SUBSTITUTION. | EXXON CHEMICAL PATENTS INC (US) | 1992-08-12 | — | — | EP | disclosed |
| EP-0220965-B1 | RESINOUS COMPOSITION CAPABLE OF RELEASING A BIOACTIVE SUBSTANCE AT A CONTROLLED RATE | Nippon Paint Co., Ltd. (JP) | 1992-01-22 | — | — | EP | disclosed |
| EP-0220965-A2 | Resinous composition capable of releasing a bioactive substance at a controlled rate | Nippon Paint Co., Ltd. (JP) | 1987-05-06 | — | — | EP | disclosed |