Dioxane

Dioxane

SCHEMBL5000306

C1COCCO1.N.O

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Dioxane. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dioxane SCHEMBL10686155 0.94
Water SCHEMBL11426218 0.94 TTR (0.86)
Dioxane SCHEMBL28845935 0.94 TTR (0.86)
Dioxane SCHEMBL305440 0.94
Dioxane SCHEMBL15882140 0.94 TTR (0.86)
Dioxane SCHEMBL23090025 0.94 TTR (0.86)
Dioxane SCHEMBL103807 0.94
Water SCHEMBL9161357 0.94 TTR (0.86)
Water SCHEMBL1866439 0.94 TTR (0.86)
Dioxane SCHEMBL2832209 0.94 TTR (0.86)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11787833-B2 Modified cyclic dinucleoside compounds as sting modulators ALIGOS THERAPEUTICS, INC. (US) 2023-10-17 US disclosed
CN-115843299-A Synthesis of oligonucleotides and related compounds 詹森生物制药有限公司 2023-03-24 CN disclosed
CN-111479813-B Triazolobenzazepines as vasopressin V1A receptor antagonists 吉瑞工厂 2023-03-21 CN disclosed
EP-3966222-A1 MODIFIED CYCLIC DINUCLEOSIDE COMPOUNDS AS STING MODULATORS Aligos Therapeutics, Inc. (US) 2022-03-16 EP disclosed
CN-114127082-A Modified cyclic dinucleoside compounds as STING modulators 阿里戈斯治疗公司 2022-03-01 CN disclosed
US-20200369711-A1 MODIFIED CYCLIC DINUCLEOSIDE COMPOUNDS AS STING MODULATORS ALIGOS THERAPEUTICS, INC. 2020-11-26 US disclosed
WO-2020227421-A1 MODIFIED CYCLIC DINUCLEOSIDE COMPOUNDS AS STING MODULATORS ALIGOS THERAPEUTICS, INC. (US) 2020-11-12 WO disclosed
CN-110023302-A 2,4, 5-trisubstituted 1,2, 4-triazolones as DHODH inhibitors 拜耳股份有限公司 2019-07-16 CN disclosed
CN-109096321-A A kind of preparation method of deoxyguanosine class organic synthesis intermediate 中国医学科学院放射医学研究所 2018-12-28 CN disclosed
CN-108467369-A BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS 诺华股份有限公司 2018-08-31 CN disclosed
US-5231174-A 2'isodideoxy-β-D-nucleosides as stable antiviral agents UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 1993-07-27 US disclosed
US-5204455-A Monomethoxytrityl protected oligonucleotides bound to a solid support ISIS PHARMACEUTICALS, INC. 1993-04-20 US disclosed
US-5164491-A Large scale synthesis of oligonucleotides and their associated analogs GILEAD SCIENCES (US) 1992-11-17 US disclosed
US-5084445-A Viricide used in treatment of AIDS UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1992-01-28 US disclosed
EP-0361831-B1 ANTIVIRAL NUCLEOSIDE COMBINATION THE WELLCOME FOUNDATION LIMITED (GB) 1992-01-22 EP disclosed
US-5077279-A Treating AIDS UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1991-12-31 US disclosed
WO-1990014831-A2 3'-AZIDO-2',3'-DIDEOXY-5-METHYLCYTIDINE ANTI-VIRAL COMPOSITION UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1990-12-13 WO disclosed
EP-0361831-A1 Antiviral nucleoside combination THE WELLCOME FOUNDATION LIMITED (GB) 1990-04-04 EP disclosed
EP-0163405-A2 Method of rate enhancement for triester synthesis of oligonucleotides using a catalytic alcohol, and compounds for use therein GENENTECH, INC. (US) 1985-12-04 EP disclosed
US-4180565-A ANTIBACTERIAL AGENTS, ANTIBIOTICS SCHERING CORPORATION (US) 1979-12-25 US disclosed