SCHEMBL5050237

SCHEMBL5050237

CC(C#N)CCC(=O)[O-].CC(C#N)CCC(=O)[O-].[Na+].[Na+]

nearest known ligand 0.58

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA1 known ✓ P00915 4/20 0.58
CA2 known ✓ P00918 3/20 0.41
BBOX1 O75936 2/20 0.47
TSHR P16473 1/20 0.43
FFAR3 O14843 2/20 0.41
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
GPR84 Q9NQS5 1/20 0.40
NFKB1 P19838 1/20 0.37
FOLH1 Q04609 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6680256 1.00 CA1 (0.58) CA1BBOX1TSHRCA2FFAR3
SCHEMBL4229227 0.78 MEN1 (0.39) CA1CA2HDAC3HDAC1HDAC2
Water SCHEMBL28240439 0.77 GABRP (0.50) TSHRFFAR3HDAC3HDAC1HDAC2
SCHEMBL7905759 0.77
SCHEMBL35490 0.77
SCHEMBL24083670 0.77
SCHEMBL4448500 0.76
SCHEMBL17389299 0.76
Hydrochloric Acid SCHEMBL7043007 0.76 GABRP (0.48) TSHRFFAR3HDAC3HDAC1HDAC2
SCHEMBL5050240 0.76 GABRP (0.48) TSHRFFAR3HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7318995-B2 Heating precusor to induce coalescence of polymer particles at exposed areas of coating; developing by applying a gum solution, removing non-exposed areas of coating from support AGFA GRAPHICS NV (BE) 2008-01-15 US disclosed
EP-1642714-B1 Method of making a negative-working lithographic printing plate. AGFA GRAPHICS NV (BE) 2007-10-24 EP disclosed
US-20060073418-A1 Heating precusor to induce coalescence of polymer particles at exposed areas of coating; developing by applying a gum solution, removing non-exposed areas of coating from support AGFA-GEVAERT (BE) 2006-04-06 US disclosed
EP-1642714-A1 Method of making a negative-working lithographic printing plate. Agfa-Gevaert (BE) 2006-04-05 EP disclosed