SCHEMBL5452840

SCHEMBL5452840

O=[N+]([O-])c1cc(S(=O)(=O)O)ccc1Cl.[Na+]

nearest known ligand 0.67

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 17/20 0.67
NPBWR1 P48145 1/20 0.60
MCHR1 Q99705 1/20 0.60
ALDH1A1 P00352 2/20 0.55
HPGD P15428 1/20 0.55
TDP1 Q9NUW8 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL332971 0.98 VCAM1 (0.69) VCAM1NPBWR1MCHR1ALDH1A1HPGD
SCHEMBL3294854 0.98 VCAM1 (0.69) VCAM1NPBWR1MCHR1ALDH1A1HPGD
SCHEMBL9585859 0.96 VCAM1 (0.67) VCAM1NPBWR1MCHR1ALDH1A1HPGD
SCHEMBL176739 0.96 VCAM1 (0.67) VCAM1NPBWR1MCHR1ALDH1A1HPGD
Hydrochloric Acid SCHEMBL6781152 0.96 VCAM1 (0.67) VCAM1NPBWR1MCHR1ALDH1A1HPGD
SCHEMBL5925286 0.84 MMP1 (0.68) VCAM1NPBWR1MCHR1ALDH1A1HPGD
SCHEMBL176738 0.84 VCAM1 (0.69) VCAM1NPBWR1MCHR1ALDH1A1
SCHEMBL10452716 0.83 VCAM1 (0.73) VCAM1NPBWR1MCHR1ALDH1A1
SCHEMBL29780388 0.83 VCAM1 (0.73) VCAM1NPBWR1MCHR1ALDH1A1
SCHEMBL809482 0.83 VCAM1 (0.73) VCAM1NPBWR1MCHR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070185176-A1 Heparanase inhibitors and uses thereof INSIGHT BIOHARMACEUTICALS LTD. (IL) 2007-08-09 US disclosed
US-5599639-A Acid-modified polybenzimidazole fuel cell elements HOECHST CELANESE CORPORATION (US) 1997-02-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070185176-A1 Heparanase inhibitors and uses thereof HPSE, ENGASE, HEXA VCAM1 540/4885NPBWR1 3521/4885MCHR1 3499/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.