SCHEMBL5480355

SCHEMBL5480355

Cc1ccccc1N1CN(S(=O)(=O)c2ccc(N)cc2)CCC1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.48
MCOLN3 Q8TDD5 1/20 0.48
HSD11B1 P28845 1/20 0.45
GAA P10253 1/20 0.45
PKM P14618 3/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
CA7 P43166 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MMP2 P08253 1/20 0.41
AKR1C3 P42330 1/20 0.41
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
HTR6 P50406 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5482778 0.86 PARL (0.47) LMNAMCOLN3HSD11B1GAAMAPK1
SCHEMBL11507468 0.78 LMNA (0.78) LMNAMCOLN3HSD11B1GAAPKM
Hydrochloric Acid SCHEMBL5474134 0.75 P2RX7 (0.45) LMNADDB1CRBN
SCHEMBL30858424 0.73 DDB1 (0.64) MEN1KMT2ADDB1CRBN
SCHEMBL5480340 0.71 P2RX7 (0.49) LMNAMEN1KMT2ADDB1CRBN
SCHEMBL6559970 0.68 KMT2A (0.56) PKMTSHRMEN1KMT2AMMP2
SCHEMBL5480222 0.68 POLB (0.57) LMNAGAAMAPK1MEN1KMT2A
SCHEMBL11306227 0.67 PKM (0.69) PKMTSHRHTTMEN1KMT2A
SCHEMBL20389408 0.67 KMT2A (0.77) GAATSHRMAPK1MEN1KMT2A
SCHEMBL1901693 0.67 DDB1 (0.56) LMNATSHRHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070010529-A1 Nitrogenous heterocyclic compounds and medical use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-01-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070010529-A1 Nitrogenous heterocyclic compounds and medical use thereof MAPK1, NOS1, NOS2 LMNA 2404/4885MCOLN3 3947/4885HSD11B1 404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.