SCHEMBL5515317

SCHEMBL5515317

CCOC(C)=C(C(C)=O)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
LMNA P02545 1/20 0.46
HSD17B10 Q99714 1/20 0.46
GLO1 Q04760 1/20 0.40
ALOX15 P16050 1/20 0.39
MGAM O43451 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
SOAT1 P35610 1/20 0.39
HCAR2 Q8TDS4 1/20 0.37
TRPA1 O75762 1/20 0.36
CYP2D6 P10635 2/20 0.33
TSHR P16473 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
MAPT P10636 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16418222 1.00 ALDH1A1 (0.46) ALDH1A1LMNAHSD17B10GLO1ALOX15
SCHEMBL5515313 1.00 ALDH1A1 (0.46) ALDH1A1LMNAHSD17B10GLO1ALOX15
SCHEMBL166091 0.90 ALDH1A1 (0.50) ALDH1A1LMNAHSD17B10GLO1ALOX15
SCHEMBL4519435 0.87 ALDH1A1 (0.52) ALDH1A1LMNAHSD17B10GLO1ALOX15
SCHEMBL9794499 0.84 ALDH1A1 (0.44) ALDH1A1LMNAHSD17B10GLO1ALOX15
SCHEMBL9794502 0.84 ALDH1A1 (0.44) ALDH1A1LMNAHSD17B10GLO1ALOX15
SCHEMBL23574259 0.82 ALDH1A1 (0.42) ALDH1A1LMNAHSD17B10GLO1ALOX15
SCHEMBL20476375 0.82 ALDH1A1 (0.42) ALDH1A1LMNAHSD17B10GLO1ALOX15
SCHEMBL20476376 0.82 ALDH1A1 (0.42) ALDH1A1LMNAHSD17B10GLO1ALOX15
SCHEMBL3678281 0.81 GLO1 (0.50) ALDH1A1LMNAHSD17B10GLO1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150099766-A1 Novel halogen-substituted compounds BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-04-09 US disclosed
US-8946234-B2 Halogen-substituted compounds BAYER CROPSCIENCE AG (DE) 2015-02-03 US disclosed
US-20110301181-A1 halogen-substituted compounds BAYER CROPSCIENCE AG (DE) 2011-12-08 US disclosed
US-7161024-B2 Process for the preparation and purification of 2-(alkoxyalkylidene)-3-ketoalkanoic acid esters from 3-ketoalkanoic acid esters SCHERING CORPORATION (US) 2007-01-09 US disclosed
EP-1644313-A2 PROCESS FOR THE PREPARATION AND PURIFICATION OF 2-(ALKOXYALKYLIDENE)-3-KETOALKANOIC ACID ESTERS FROM 3-KETOALKANOIC ACID ESTERS SCHERING CORPORATION (US) 2006-04-12 EP disclosed
US-20050027140-A1 Process for the preparation and purification of 2-(alkoxyalkylidene)-3-ketoalkanoic acid esters from 3-ketoalkanoic acid esters SCHERING CORPORATION 2005-02-03 US disclosed
WO-2005007608-A2 PROCESS FOR THE PREPARATION AND PURIFICATION OF 2-(ALKOXYALKYLIDENE)-3-KETOALKANOIC ACID ESTERS FROM 3-KETOALKANOIC ACID ESTERS SCHERING CORPORATION (US) 2005-01-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050027140-A1 Process for the preparation and purification of 2-(alkoxyalkylidene)-3-ketoalkanoic acid esters from 3-ketoalkanoic acid esters ACKR3, CCR5, CCRL2 ALDH1A1 437/4885LMNA 3977/4885HSD17B10 878/4885
US-20110301181-A1 halogen-substituted compounds L3MBTL4, QSOX1, L3MBTL3 ALDH1A1 457/4885LMNA 209/4885HSD17B10 3268/4885
US-20150099766-A1 Novel halogen-substituted compounds L3MBTL4, PRDX4, PRDX1 ALDH1A1 522/4885LMNA 626/4885HSD17B10 3719/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.