SCHEMBL5844904

SCHEMBL5844904

O=C(O)N(CC1C2CCC1N(Cc1ccccc1)C2)c1ccc(F)c([N+](=O)[O-])c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.38
MAPT P10636 3/20 0.38
TP53 P04637 1/20 0.38
KMT2A Q03164 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 2/20 0.38
ACHE P22303 3/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
SIGMAR1 Q99720 2/20 0.36
CFTR P13569 1/20 0.35
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM3 P20309 1/20 0.35
PTGS2 P35354 1/20 0.34
FAAH O00519 1/20 0.34
ROCK2 O75116 1/20 0.33
ARHGDIA P52565 1/20 0.33
ROCK1 Q13464 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5833003 0.85 SIGMAR1 (0.41) LMNAKMT2AALDH1A1ACHEPOLB
SCHEMBL5844908 0.81 LMNA (0.36) LMNAMAPTTP53KMT2AALDH1A1
SCHEMBL5833539 0.81 CHRM2 (0.47) MAPTSIGMAR1CHRM2CHRM3ROCK2
SCHEMBL5833452 0.78 DCUN1D1 (0.40) KMT2AMEN1ACHESIGMAR1UBE2M
SCHEMBL5833112 0.78 ROCK2 (0.41) ACHECHRM2CHRM3FAAHROCK2
SCHEMBL5833937 0.77 OPRD1 (0.47) KMT2AACHEHTTCHRM2CHRM3
SCHEMBL5833278 0.77 RNF4 (0.42) ACHECHRM2CHRM3FAAH
SCHEMBL5833269 0.77 KDM1A (0.40) KMT2AMEN1FAAHMCHR1DCUN1D1
SCHEMBL5833430 0.75 SIGMAR1 (0.43) KMT2AMEN1ACHEPOLBSIGMAR1
SCHEMBL5833024 0.74 BRD4 (0.38) KMT2AMEN1SIGMAR1CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7008955-B2 (2-azabicyclo[2.2.1]hept-7yl) methanol derivatives as nicotinic acetylcholine receptor agonists MERCK PATENT GMBH (DE) 2006-03-07 US claimed