SCHEMBL6004130

SCHEMBL6004130

c1cnc2nc(-c3csc4ccccc34)c(Oc3ccnc4ccccc34)cc2c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGK1 P00558 1/20 0.35
TGFBR1 P36897 1/20 0.35
BRAF P15056 3/20 0.34
KDR P35968 2/20 0.34
PDE10A Q9Y233 2/20 0.33
CDC7 O00311 1/20 0.33
HTR1A P08908 2/20 0.33
CYP3A4 P08684 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
MAPK14 Q16539 1/20 0.32
TNNI3K Q59H18 1/20 0.32
ERN1 O75460 1/20 0.31
TUBB4A P04350 1/20 0.31
TUBB P07437 1/20 0.31
TUBA3C P0DPH7 1/20 0.31
TUBA1B P68363 1/20 0.31
TUBA4A P68366 1/20 0.31
TUBB4B P68371 1/20 0.31
TUBB3 Q13509 1/20 0.31
TUBB2A Q13885 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6005298 0.88 SRC (0.44) PGK1TGFBR1KDR
SCHEMBL6004276 0.81 LMNA (0.39) BRAFKDRCYP3A4
SCHEMBL6004283 0.78 ERN1 (0.40) PGK1TGFBR1CDC7HTR1AERN1
SCHEMBL6004728 0.77 CYP1A2 (0.37) BRAFKDRCYP3A4MAPK14
SCHEMBL6002787 0.70 CCNC (0.39) BRAFPDE10AMAPK14
SCHEMBL6005302 0.70 DHODH (0.39) MAPK14
SCHEMBL6004327 0.69 TOP1 (0.42) MAPK14
SCHEMBL9431770 0.68 NCF1 (0.54) BRAFKDRHTR1ACYP3A4MAPK14
SCHEMBL6002953 0.68 TGFBR1 (0.41) TGFBR1PDE10A
SCHEMBL6004287 0.68 TGFBR1 (0.41) TGFBR1PDE10AERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed