SCHEMBL6004728

SCHEMBL6004728

Brc1ccc(-c2nc3ncccc3cc2Oc2ccnc3ccccc23)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
HTT P42858 1/20 0.37
KDR P35968 2/20 0.36
BRAF P15056 2/20 0.35
CYP1B1 Q16678 2/20 0.35
CYP3A4 P08684 2/20 0.35
SYK P43405 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
MAPK14 Q16539 1/20 0.33
DHODH Q02127 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004276 0.91 LMNA (0.39) KDRBRAFCYP3A4SYKLMNA
SCHEMBL6002787 0.80 CCNC (0.39) BRAFMAPK14DHODH
SCHEMBL6004327 0.79 TOP1 (0.42) KDM4ELMNAMAPK14DHODHMAPT
SCHEMBL6005302 0.79 DHODH (0.39) HTTKDM4EMAPK14DHODH
SCHEMBL6004812 0.78 FGFR2 (0.44) KDR
SCHEMBL6004803 0.77 FGFR2 (0.36) KDRDHODH
SCHEMBL6004795 0.77 FGFR2 (0.36) KDRMAPK14DHODH
SCHEMBL6004736 0.77 KDM4E (0.48) KDRCYP3A4KDM4E
SCHEMBL6005261 0.77 KDM4E (0.49) CYP1A2CYP2C19KDRCYP3A4KDM4E
SCHEMBL6004130 0.77 PGK1 (0.35) KDRBRAFCYP3A4MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed