SCHEMBL6206466

SCHEMBL6206466

O=C1CCN(c2ccc(N3CCOC3=O)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.42
KDM1A O60341 2/20 0.40
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
RCOR1 Q9UKL0 2/20 0.40
F10 P00742 2/20 0.39
CCNA2 P20248 3/20 0.37
CDK2 P24941 3/20 0.37
CCNA1 P78396 3/20 0.37
CCNB2 O95067 1/20 0.37
CCNE2 O96020 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
EP300 Q09472 1/20 0.35
KAT2B Q92831 1/20 0.35
CCNC P24863 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14810230 0.86 EP300 (0.47) TNKSEP300KAT2B
SCHEMBL8259337 0.81 ADRB1 (0.49) TNKS
SCHEMBL27620742 0.81 LGMN (0.48) TNKSKDM1AMAOAMAOBRCOR1
SCHEMBL1377738 0.78 KDM1A (0.46) TNKSKDM1AMAOAMAOBRCOR1
SCHEMBL20907468 0.77 LMNA (0.54) EP300KAT2B
SCHEMBL3584707 0.77 ALOX15 (0.37) TNKS
SCHEMBL2535607 0.77 TNKS (0.45) TNKSKDM1AMAOAMAOBRCOR1
SCHEMBL2535612 0.77 DGAT1 (0.51) TNKSKDM1AMAOAMAOBRCOR1
SCHEMBL13167913 0.77 HSD11B1 (0.47) TNKSKDM1AMAOAMAOBRCOR1
SCHEMBL1455890 0.77 BCL2 (0.48) TNKSKDM1AMAOAMAOBRCOR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1565461-A2 ANTIBACTERIAL SUBSTITUTED CYANOMETHYL(ENE)PIPERIDINOPHENYL OXAZOLIDINONES, PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Patel, Mahesh V. (IN) 2005-08-24 EP claimed
US-20040063954-A1 Antibacterial cyano-(substituted)-methylenepiperidinophenyl oxazolidinones targeting multiple ribonucleoprotein sites WOCKHARDT LIMITED 2004-04-01 US claimed
WO-2004007489-A2 ANTIBACTERIAL SUBSTITUTED CYANOMETHYL (ENE) PIPERIDINOPHENYL OXAZOLIDINONES, PROCESS OR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM WOCKHARDT LIMITED (IN) 2004-01-22 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063954-A1 Antibacterial cyano-(substituted)-methylenepiperidinophenyl oxazolidinones targeting multiple ribonucleoprotein sites POLRMT, RNASEL, RNASE1 TNKS 701/4885KDM1A 2142/4885MAOA 1873/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.